Target Details
| UniProt AC | Q96L34 |
|---|---|
| Gene Symbol | MARK4 |
| Protein Name | MAP/microtubule affinity-regulating kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 43
- Clinical molecules 10
- Avg pChEMBL 7.12
Active Molecules (43)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.6 | IC50 | 408 | — | |
OWRXHGAFWZFFCW
|
9.3 | Ki | 113 | — | |
HKSZLNNOFSGOKW
|
9.1 | Ki | 118 | — | |
OFIFLUFVENTCNZ
|
8.7 | IC50 | 11 | — | |
HKSZLNNOFSGOKW
|
8.3 | Kd | 213 | — | |
NXSJMRCTGYTSTK
|
8.2 | Kd | 200 | — | |
LRZYYIZFBXFSJB
|
8.1 | Ki | 69 | — | |
PBCZSGKMGDDXIJ
|
8.1 | Kd | 68 | Yes | |
RYYNGWLOYLRZLK
|
8.1 | Kd | 45 | — | |
QQWUGDVOUVUTOY
|
7.9 | Kd | 231 | Yes | |
XLFNLJYGUOLEJS
|
7.7 | IC50 | 26 | — | |
DYNHJHQFHQTFTP
|
7.6 | Kd | 38 | — | |
KOZFSFOOLUUIGY
|
7.5 | Kd | 88 | Yes | |
AYCPARAPKDAOEN
|
7.5 | Kd | 73 | — | |
YFNWWNRZJGMDBR
|
7.4 | Kd | 35 | — | |
ZSZOBRBJIJWWHH
|
7.1 | IC50 | 4 | — | |
PRRYQINUAIQTFJ
|
7.1 | Ki | 11 | — | |
ZCCPLJOKGAACRT
|
7.1 | Kd | 599 | — | |
MZDKLVOWGIOKTN
|
7.1 | Kd | 80 | — | |
NHHQJBCNYHBUSI
|
7.0 | Kd | 220 | — | |
UIARLYUEJFELEN
|
6.9 | Kd | 289 | Yes | |
OPSONJKOCBCHTM
|
6.7 | IC50 | 2 | — | |
YYLKKYCXAOBSRM
|
6.7 | Kd | 191 | — | |
IOYFYUOBKSQTFF
|
6.7 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
6.6 | Kd | 64 | Yes | |
JZTOUVBEZONDKA
|
6.6 | Ki | 80 | — | |
UHEQNWGXIQUUOV
|
6.6 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.5 | Kd | 137 | Yes | |
UKBGBACORPRCGG
|
6.5 | IC50 | 17 | — | |
DMMILYKXNCVKOJ
|
6.5 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.4 | Kd | 91 | Yes | |
OUJZYQBEFNDJQN
|
6.4 | Ki | 71 | — | |
UYJNQQDJUOUFQJ
|
6.4 | Ki | 68 | — | |
NLYZJYHBZFQGDP
|
6.3 | IC50 | 2 | — | |
IAYGCINLNONXHY
|
6.3 | Kd | 50 | — | |
YQKQQLKFPBCSDP
|
6.3 | IC50 | 2 | — | |
APKZTNIHDKUHTG
|
6.3 | IC50 | 2 | — | |
UJLAWZDWDVHWOW
|
6.2 | Ki | 11 | — | |
KDKUVYLMPJIGKA
|
6.2 | Kd | 91 | Yes | |
LOZGENZISGZHOI
|
6.0 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.0 | Kd | 139 | — | |
GCIKSSRWRFVXBI
|
6.0 | Ki | 109 | Yes |