Target Details
| UniProt AC | Q96KQ7 |
|---|---|
| Gene Symbol | EHMT2 |
| Protein Name | Histone-lysine N-methyltransferase EHMT2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 185
- Clinical molecules 1
- Avg pChEMBL 7.05
KEGG Pathways (3)
Active Molecules (185)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBKLIARRJUTMTQ
|
6.3 | IC50 | 7 | — | |
PYGWCVPYKMILCJ
|
6.3 | IC50 | 2 | — | |
WLSUJPBXUGENOU
|
6.3 | IC50 | 2 | — | |
MLTCNEHPZTWJKH
|
6.3 | IC50 | 2 | — | |
YQVURWXJUBXXCZ
|
6.3 | IC50 | 2 | — | |
FIVPIPIDMRVLAY
|
6.3 | IC50 | 7 | Yes | |
GDWIBPWOSOTLGZ
|
6.3 | IC50 | 2 | — | |
GRCRJEGHKCSKNE
|
6.3 | IC50 | 2 | — | |
UWTQREDSTMKGMT
|
6.3 | IC50 | 2 | — | |
KUAZQDVKQLNFPE
|
6.3 | IC50 | 9 | — | |
LNLYAENQQBUQGQ
|
6.3 | IC50 | 2 | — | |
YWWZCHLUQSHMCL
|
6.3 | IC50 | 2 | — | |
ZJUKTBDSGOFHSH
|
6.2 | Ki | 22 | — | |
FKTQPAVLUZRKHC
|
6.2 | IC50 | 2 | — | |
AUZONCFQVSMFAP
|
6.2 | IC50 | 15 | — | |
BBJDFTWFOONSLK
|
6.2 | IC50 | 2 | — | |
PVVLIIZIQXDFSP
|
6.2 | IC50 | 2 | — | |
CUXOFABLNDVFGR
|
6.2 | IC50 | 2 | — | |
MDFCEIJITSVGGO
|
6.2 | IC50 | 2 | — | |
YYFDMPHIONBOKZ
|
6.2 | IC50 | 3 | — | |
KNLMZFKJTDDDQH
|
6.2 | Ki | 3 | — | |
SXUDOJDVYKVXEH
|
6.2 | IC50 | 2 | — | |
LSNVRHZIUYXNRN
|
6.1 | IC50 | 2 | — | |
OPOCBCGSTOFGIL
|
6.1 | IC50 | 2 | — | |
SEIITEYCJLDVFW
|
6.1 | IC50 | 2 | — | |
GQJJJDCHUVVIMA
|
6.1 | IC50 | 2 | — | |
AKOSZLHLQSSJQB
|
6.1 | IC50 | 2 | — | |
JBMUWBUCVSKHLE
|
6.1 | Kd | 2 | — | |
ZYNUWSFRZCRKSN
|
6.1 | IC50 | 2 | — | |
RUPLHSKMNNTYKA
|
6.1 | IC50 | 2 | — | |
ZDTIJWKWNYJIAB
|
6.1 | IC50 | 2 | — | |
NEJODHSPAWSHOK
|
6.0 | IC50 | 2 | — | |
XLDKAPYGJVCXCU
|
6.0 | IC50 | 2 | — | |
YMSMSNAIHUSOEZ
|
6.0 | IC50 | 2 | — | |
FNDUCTFWOZQGTB
|
6.0 | IC50 | 2 | — |