Target Details
| UniProt AC | Q96KQ7 |
|---|---|
| Gene Symbol | EHMT2 |
| Protein Name | Histone-lysine N-methyltransferase EHMT2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 185
- Clinical molecules 1
- Avg pChEMBL 7.05
KEGG Pathways (3)
Active Molecules (185)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BYCFGRRIIUNHIZ
|
6.7 | IC50 | 2 | — | |
CHEFNBAYIGSOIR
|
6.7 | IC50 | 3 | — | |
RWIWOWGXKHFTHM
|
6.7 | IC50 | 2 | — | |
WGTLTEYVKMNATO
|
6.7 | IC50 | 2 | — | |
KGUAKPWBXICIMX
|
6.7 | IC50 | 2 | — | |
VAAQORJZPYRYHH
|
6.7 | IC50 | 2 | — | |
CHOFEGBVNPOIOH
|
6.7 | IC50 | 2 | — | |
KZOJJUVZAJGNQV
|
6.6 | IC50 | 2 | — | |
KKXRBRPMTQSNTJ
|
6.6 | IC50 | 3 | — | |
PCKQRGGTJLXKRR
|
6.6 | IC50 | 2 | — | |
YBQHFHPOKHPBRB
|
6.6 | IC50 | 2 | — | |
VWFQZXWQZKXLEI
|
6.6 | IC50 | 2 | — | |
BZYQCFUKLXJLGU
|
6.6 | IC50 | 5 | — | |
ZBCTVJOKADNKNK
|
6.6 | IC50 | 4 | — | |
DJKVIUVJRXEKNV
|
6.5 | IC50 | 2 | — | |
DUFHUIJOFOYTAR
|
6.5 | IC50 | 2 | — | |
FWANMJZHBHKDKO
|
6.5 | IC50 | 2 | — | |
RDXCLLLMCWXDJB
|
6.5 | IC50 | 2 | — | |
ZNNQDTNCHFJGMI
|
6.5 | IC50 | 2 | — | |
MBUONUPUCSDIFQ
|
6.5 | IC50 | 2 | — | |
MROKTUUFAWVTEF
|
6.5 | IC50 | 2 | — | |
NEHZFWWDTWSDKX
|
6.5 | IC50 | 2 | — | |
AFFYALXSRBVAPQ
|
6.5 | IC50 | 2 | — | |
PGVIWADEDHEJGB
|
6.5 | IC50 | 2 | — | |
PZFSXMLFZTZWAI
|
6.5 | IC50 | 2 | — | |
RINVPEJSDRLKKC
|
6.5 | IC50 | 2 | — | |
AUGGZTSGLVEWLK
|
6.5 | IC50 | 2 | — | |
YYXVQDZRELJUBX
|
6.5 | IC50 | 2 | — | |
FKRRYTPCUFOKGU
|
6.5 | IC50 | 2 | — | |
NKRNUYLZAXRLJU
|
6.5 | IC50 | 2 | — | |
YTZXLVDHUCDBOG
|
6.5 | IC50 | 2 | — | |
IQRVFHPCSDGBCR
|
6.5 | IC50 | 2 | — | |
MPYDHWGOMXNQOW
|
6.5 | IC50 | 2 | — | |
AVSMKKGLVDCOEU
|
6.5 | IC50 | 2 | — | |
NDEREOOBAVLGBN
|
6.5 | IC50 | 2 | — | |
DTBKCXDRYUDIPI
|
6.4 | IC50 | 2 | — | |
JIPXEHIHQRXFCZ
|
6.4 | IC50 | 2 | — | |
SJSJYFGBZRKJLV
|
6.4 | IC50 | 2 | — | |
RCWUUMJJJVFQSV
|
6.4 | IC50 | 2 | — | |
DYEFUKCXAQOFHX
|
6.4 | IC50 | 31 | — | |
WGURLEOJEIDTBP
|
6.4 | IC50 | 2 | — | |
CXHSPDIJBBFXBC
|
6.4 | IC50 | 2 | — | |
PIXKGBJULNYOEX
|
6.4 | IC50 | 2 | — | |
MEVMMQQJOXBSAX
|
6.3 | IC50 | 2 | — | |
RBBZOCOZIYNTCM
|
6.3 | IC50 | 2 | — | |
TYZFQSLJTWPSDS
|
6.3 | IC50 | 2 | — | |
XZUWJVJVVBARGQ
|
6.3 | IC50 | 2 | — | |
YRFPHJAMBMALTM
|
6.3 | IC50 | 2 | — | |
AMAQJTHMSLYMFT
|
6.3 | IC50 | 2 | — | |
GLDHWRNHMTWDKJ
|
6.3 | IC50 | 2 | — |