Target Details
| UniProt AC | Q96KQ7 |
|---|---|
| Gene Symbol | EHMT2 |
| Protein Name | Histone-lysine N-methyltransferase EHMT2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 185
- Clinical molecules 1
- Avg pChEMBL 7.05
KEGG Pathways (3)
Active Molecules (185)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LZYFRBDZTMNLFR
|
7.6 | IC50 | 4 | — | |
OWORSODZTADOQX
|
7.6 | IC50 | 2 | — | |
XAHHWLRJWBHPFE
|
7.5 | IC50 | 2 | — | |
AUFSXIYCIRDGIZ
|
7.5 | IC50 | 2 | — | |
NYDFIFBPOWTDSS
|
7.5 | IC50 | 2 | — | |
ZAGKOOCPARJINO
|
7.5 | IC50 | 2 | — | |
WTVIBMHPUDQIBD
|
7.5 | IC50 | 3 | — | |
GWLDWJBHEXGGHH
|
7.4 | IC50 | 2 | — | |
KXENQCUVSMIIGA
|
7.4 | IC50 | 2 | — | |
QMIDRDYKZINKHP
|
7.4 | IC50 | 2 | — | |
YNEOJEHDXDSCBD
|
7.4 | IC50 | 2 | — | |
PZPUORZZMLOXMT
|
7.4 | IC50 | 2 | — | |
ABOYMKZJGPBYCR
|
7.3 | IC50 | 2 | — | |
JKEZOPHKGXCQKI
|
7.3 | IC50 | 4 | — | |
BRSOLPMHTWMRJJ
|
7.3 | IC50 | 4 | — | |
ZDINBSHEURZXDD
|
7.3 | IC50 | 2 | — | |
GWWFCFPTRJUJIM
|
7.3 | IC50 | 2 | — | |
QOECJCJVIMVJGX
|
7.3 | IC50 | 8 | — | |
ZFYXXFFBVZGXLX
|
7.3 | IC50 | 2 | — | |
VDFCTSUFEJCENU
|
7.3 | IC50 | 2 | — | |
OQXGDFSYMGTLHG
|
7.3 | IC50 | 7 | — | |
AEJULKFUIXWPOX
|
7.2 | IC50 | 2 | — | |
FWEMDGGXZBEQDX
|
7.2 | IC50 | 2 | — | |
DCCAQKTZHJSEKP
|
7.2 | IC50 | 2 | — | |
MJGRJTGEKSYWOA
|
7.1 | IC50 | 2 | — | |
AHSGGTMURLDJJM
|
7.1 | IC50 | 2 | — | |
PUCHZOBUKOKFRK
|
7.1 | IC50 | 2 | — | |
GKNHULHXRNRLNS
|
7.0 | IC50 | 2 | — | |
GOCBKOQITCNXIM
|
7.0 | IC50 | 2 | — | |
KJOYGBHVQOPLES
|
7.0 | IC50 | 2 | — | |
FGAGTVKUPJXOMV
|
7.0 | IC50 | 2 | — | |
FNRUPVONTWZCGL
|
7.0 | IC50 | 2 | — | |
LDFAJFPHFKEJOI
|
7.0 | IC50 | 2 | — | |
LMXOHSDXUQEUSF
|
7.0 | IC50 | 6 | — | |
FNKMWVAWPMHKHA
|
7.0 | IC50 | 2 | — | |
KLWZLAHWDCVBRC
|
7.0 | IC50 | 2 | — | |
RNAMYOYQYRYFQY
|
7.0 | IC50 | 3 | — | |
NZIRMQGNRYJHOB
|
6.9 | IC50 | 2 | — | |
IVTVGDXNLFLDRM
|
6.9 | IC50 | 8 | — | |
AJHIQURHJXOCCP
|
6.9 | IC50 | 2 | — | |
STWMZHHKHUOUQD
|
6.9 | IC50 | 2 | — | |
OSXFATOLZGZLSK
|
6.9 | IC50 | 3 | — | |
GWCXSYHLYREIAK
|
6.8 | IC50 | 2 | — | |
FDUSNRNFGPEONK
|
6.8 | IC50 | 2 | — | |
LHNQVGYVOOWUCA
|
6.8 | IC50 | 2 | — | |
DCGOBPRQIYFVOD
|
6.8 | IC50 | 2 | — | |
SFOCRSFKWQNGAT
|
6.8 | IC50 | 2 | — | |
ZRZWBWPDBOVIGQ
|
6.8 | IC50 | 4 | — | |
CZXPVZMKOLPPPQ
|
6.8 | IC50 | 2 | — | |
LNFNHVCQOOPPAK
|
6.7 | IC50 | 2 | — |