Target Details
| UniProt AC | Q96KQ7 |
|---|---|
| Gene Symbol | EHMT2 |
| Protein Name | Histone-lysine N-methyltransferase EHMT2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00023 (Ank) PF12796 (Ank_2) PF21533 (EHMT1-2_CRR) PF05033 (Pre-SET) PF00856 (SET) |
Summary
- Multi-target molecules 185
- Clinical molecules 1
- Avg pChEMBL 7.05
KEGG Pathways (3)
Active Molecules (185)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WOXWYMQYSSZYNQ
|
9.3 | IC50 | 2 | — | |
FQOJFAZVDGPADJ
|
9.2 | IC50 | 3 | — | |
FACDBZNPDREQDS
|
8.7 | IC50 | 2 | — | |
WXSNAPMHXWGVRQ
|
8.7 | IC50 | 2 | — | |
CVWPNABDQLFDLZ
|
8.5 | IC50 | 2 | — | |
SKDSVUVJPWHTOI
|
8.5 | IC50 | 2 | — | |
USIHDOVZZRFRAY
|
8.5 | IC50 | 2 | — | |
BKCDJTRMYWSXMC
|
8.5 | IC50 | 3 | — | |
UQBQMWLGFSNAIR
|
8.5 | IC50 | 2 | — | |
ZVPMIOYZZZPGFF
|
8.4 | IC50 | 4 | — | |
JOHUZOVWSNNWQZ
|
8.4 | IC50 | 2 | — | |
JWHZKAWJXRZCOW
|
8.3 | IC50 | 2 | — | |
DKHFXUKOWLZXHX
|
8.2 | IC50 | 2 | — | |
QUDNDJNGIQINLE
|
8.2 | IC50 | 2 | — | |
QYKHEFBHQZYBTF
|
8.2 | IC50 | 2 | — | |
VUIKWDIDFZKLCE
|
8.2 | IC50 | 2 | — | |
MFOQRJHECLPWDG
|
8.2 | IC50 | 2 | — | |
NDKARMJRFVQCIS
|
8.2 | IC50 | 2 | — | |
GXAJALCTHNRXSM
|
8.2 | IC50 | 2 | — | |
PCZXRYSXMPNRDU
|
8.2 | IC50 | 2 | — | |
LMGRXYCLENIEMO
|
8.1 | IC50 | 3 | — | |
QHYRXLJGNSPRGA
|
8.1 | IC50 | 2 | — | |
RLQLKZTYUYIWDB
|
8.1 | IC50 | 2 | — | |
GHCDVBSKNGUGCK
|
8.1 | IC50 | 2 | — | |
AULLUGALUBVBDD
|
8.1 | IC50 | 2 | — | |
RJXNYIVGMQXAMD
|
8.0 | IC50 | 2 | — | |
QAQNPAOMUGDFRD
|
8.0 | IC50 | 2 | — | |
RDPYODVIYQQQFZ
|
8.0 | IC50 | 2 | — | |
KUEVRQLZRITNEE
|
7.9 | IC50 | 2 | — | |
VMVRYCYPSDCNEH
|
7.9 | IC50 | 2 | — | |
UNRCZHRRDXQTEH
|
7.9 | IC50 | 2 | — | |
ZAWYCUBKBPHGBY
|
7.9 | IC50 | 2 | — | |
SJRUKFZRLQHAEM
|
7.8 | IC50 | 2 | — | |
YBKZQRANOVULPZ
|
7.8 | IC50 | 2 | — | |
JHSAFANTCQXEFJ
|
7.8 | IC50 | 2 | — | |
KBLFJYYDDWJDKG
|
7.8 | IC50 | 2 | — | |
ONQXWOCNSKDACO
|
7.8 | IC50 | 2 | — | |
UDDYBHJZHUMVFR
|
7.8 | IC50 | 2 | — | |
UUFAYOSBAHOCOU
|
7.8 | IC50 | 2 | — | |
XIVUGRBSBIXXJE
|
7.8 | IC50 | 2 | — | |
ZZSNUOGALFUINV
|
7.8 | IC50 | 2 | — | |
VMMRDFLDWHFNOX
|
7.8 | IC50 | 4 | — | |
HWEQZXCORSHBDW
|
7.8 | IC50 | 2 | — | |
PQJVPCANHLGIOZ
|
7.7 | IC50 | 2 | — | |
RXNZKWRSWQWERQ
|
7.7 | IC50 | 2 | — | |
HXTSAISPABOHHN
|
7.7 | IC50 | 2 | — | |
UOHZNWFNUIYUCY
|
7.7 | IC50 | 2 | — | |
YNISGSVZVOGISR
|
7.7 | IC50 | 2 | — | |
BIJYNDLTSDYKHJ
|
7.7 | IC50 | 2 | — | |
DATFGAXLCSNDRI
|
7.6 | IC50 | 2 | — |