Target Details
| UniProt AC | Q96KB5 |
|---|---|
| Gene Symbol | PBK |
| Protein Name | Lymphokine-activated killer T-cell-originated protein kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 247
- Clinical molecules 1
- Avg pChEMBL 7.87
Active Molecules (247)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LHZSCNHIQYURJR
|
7.2 | IC50 | 2 | — | |
UISKFSKGRDJBFK
|
7.2 | IC50 | 2 | — | |
BAGJPDYVOWKTFN
|
7.2 | IC50 | 2 | — | |
QSTRDZKAPUTJCL
|
7.2 | IC50 | 2 | — | |
IVTXKZOAEFIJGG
|
7.2 | IC50 | 2 | — | |
INSXCHLFWDLFGN
|
7.2 | IC50 | 2 | — | |
CAQDNIUJCQIJSN
|
7.2 | IC50 | 2 | — | |
MBWJUWFANMBYHY
|
7.2 | IC50 | 2 | — | |
HKKPCLDSLIZWJM
|
7.1 | IC50 | 2 | — | |
APIJSFSFSPDPLN
|
7.1 | IC50 | 2 | — | |
OUVMMTWUDVNCFP
|
7.1 | IC50 | 2 | — | |
QBTAZLWMEYVBSX
|
7.1 | IC50 | 2 | — | |
VUEWLORAHCWFHP
|
7.1 | IC50 | 2 | — | |
MMYHBULUVREXPP
|
7.1 | IC50 | 2 | — | |
LGICPSFBCIDMAT
|
7.1 | IC50 | 2 | — | |
OIOUIPSTQHPGEN
|
7.1 | IC50 | 2 | — | |
DNRFMSJVTXHVCU
|
7.1 | IC50 | 2 | — | |
SJVBKIJJPQBWCC
|
7.1 | IC50 | 2 | — | |
JOYSKMLFEFBTPY
|
7.1 | IC50 | 2 | — | |
YKNNQNCGYOGHRS
|
7.0 | IC50 | 2 | — | |
XCFRUAOZMVFDPQ
|
7.0 | IC50 | 2 | — | |
FPQHXFMYXQZPSV
|
6.7 | Ki | 23 | — | |
UTFXYGYVDDLJER
|
6.6 | Ki | 36 | — | |
DJUSDFVEBBYFFL
|
6.5 | Ki | 27 | — | |
GUHUQPHEGAYGKK
|
6.5 | Ki | 4 | — | |
UUYUVYXSHUTRGO
|
6.5 | Ki | 4 | — | |
MWKSRKSEWLRPBL
|
6.4 | Kd | 1075 | — | |
CZIGMBNEFWBEMD
|
6.4 | Ki | 16 | — | |
FQEODTMNWMDUMD
|
6.4 | Ki | 25 | — | |
GHAZVJQMLWOQLP
|
6.4 | Ki | 17 | — | |
OWDRQHVEJIYVOI
|
6.4 | Ki | 47 | — | |
YKJSWMAVAKRUAN
|
6.4 | Ki | 19 | — | |
BSFNGHCTZDCQBF
|
6.3 | Ki | 93 | — | |
DBKQWGCVGCVPIP
|
6.3 | Ki | 21 | — | |
DKXHSOUZPMHNIZ
|
6.3 | Ki | 51 | Yes | |
SGHXFHRRWFLILP
|
6.3 | Ki | 29 | — | |
XBDWKVLCDCUNHH
|
6.3 | Ki | 18 | — | |
ADMFLILDQJSEIK
|
6.2 | Ki | 72 | — | |
DFMCXVONDDGQIY
|
6.2 | Ki | 66 | — | |
GUMBHNMWKMFKRT
|
6.2 | Ki | 23 | — | |
NLUPJKQOKWBWFC
|
6.2 | Ki | 69 | — | |
XPHWIERLJBFPFV
|
6.2 | Ki | 69 | — | |
DBXGGXLBTWZXBB
|
6.1 | Ki | 39 | — | |
OLVBAUVSICCWEJ
|
6.1 | Ki | 39 | — | |
PAIFYAZSILXLBO
|
6.1 | Ki | 26 | — | |
KRIUNPBAQZGFQA
|
6.0 | Ki | 76 | — | |
YWTBGJGMTBHQTM
|
6.0 | Ki | 65 | — |