Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MBKBRIBQHFBRHO
|
8.4 | IC50 | 3 | — | |
MBKBRIBQHFBRHO
|
8.4 | IC50 | 3 | — | |
MSGWNYXBVMCUNQ
|
8.4 | IC50 | 3 | — | |
NDJAPUTXCKBOMQ
|
8.4 | IC50 | 2 | — | |
NFYDBBVZKANMEX
|
8.4 | IC50 | 4 | — | |
OPVKJVDDNDEKSB
|
8.4 | IC50 | 2 | — | |
PSWIPMICOQJHRP
|
8.4 | IC50 | 3 | — | |
QJOLFMLQXIPTTF
|
8.4 | IC50 | 3 | — | |
QONPPIZSNSSCSK
|
8.4 | Ki | 45 | Yes | |
RBMOLIOJAWRTIV
|
8.4 | IC50 | 4 | — | |
RJTVPQLMBWIFKC
|
8.4 | IC50 | 5 | — | |
SRUYMJRFVGLQDV
|
8.4 | Ki | 37 | — | |
VEJCMMPVTMQFME
|
8.4 | Ki | 8 | Yes | |
WKKLEERAKHQFTN
|
8.4 | IC50 | 3 | — | |
ZFQFDCSTGATGQP
|
8.4 | IC50 | 4 | — | |
ZLODPJRHCQWJSX
|
8.4 | IC50 | 3 | — | |
ZNZJOKVVRNTGRH
|
8.4 | IC50 | 2 | — | |
ZZFGCFQOWNBGHP
|
8.4 | IC50 | 2 | — | |
MAZAMYSGSCRKQA
|
8.4 | IC50 | 3 | — | |
VHNNKJCKILGDNA
|
8.4 | IC50 | 5 | — | |
GWQXSFUEKBLIOK
|
8.4 | IC50 | 3 | — | |
BRXIQCXGFZUJEE
|
8.4 | IC50 | 3 | — | |
KCMYPBPMTXEKNF
|
8.4 | IC50 | 7 | — | |
MFRRIEBIBJQMAF
|
8.4 | IC50 | 3 | — | |
DIZTWKKXOXSRQF
|
8.4 | IC50 | 2 | — | |
SMOTZGTWZKCZAR
|
8.4 | IC50 | 2 | — | |
WPSTUURUTXEJCF
|
8.4 | IC50 | 3 | — | |
KRUKDVBCEQTOCL
|
8.3 | IC50 | 3 | — | |
YXVZSMQKDLURNT
|
8.3 | IC50 | 3 | Yes | |
LCVIRAZGMYMNNT
|
8.3 | IC50 | 4 | — | |
NQOIWUCLZREOSK
|
8.3 | IC50 | 2 | — | |
OPVKJVDDNDEKSB
|
8.3 | IC50 | 2 | — | |
XISIJMIPHPQCQQ
|
8.3 | IC50 | 9 | — | |
CMWCUAWBNRSCEK
|
8.3 | IC50 | 3 | Yes | |
DWMNINPORGJSKR
|
8.3 | IC50 | 3 | Yes | |
ICODOOXDNPOINQ
|
8.3 | IC50 | 3 | — | |
QQCDNHWVJDMTCC
|
8.3 | IC50 | 2 | — | |
SIDSSTAVUKNHFG
|
8.3 | IC50 | 2 | — | |
BCSHETJKMWOYNN
|
8.3 | IC50 | 2 | — | |
BQWUBCRDJPIJAT
|
8.3 | Ki | 10 | — | |
CCCMIDUAEDVYME
|
8.3 | IC50 | 3 | Yes | |
CPGPEVNIOCXOPN
|
8.3 | IC50 | 3 | — | |
CQBBMNXXVMOFCA
|
8.3 | Ki | 39 | — | |
DINLHKGZVRGQQO
|
8.3 | IC50 | 3 | — | |
GCHPTPVYEQUDIU
|
8.3 | IC50 | 2 | — | |
IDAYTJFWXHMPGK
|
8.3 | Ki | 3 | — | |
JXCWQMODNUZVKT
|
8.3 | IC50 | 3 | — | |
LNYPORVAHOFKGG
|
8.3 | Ki | 3 | — | |
NKRSLISCOPHPJT
|
8.3 | IC50 | 3 | — | |
OIUQFNNWKMANNS
|
8.3 | IC50 | 3 | — |