Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORAPIBKWDRGVHK
|
8.5 | IC50 | 2 | — | |
OTACRQCAOBRLAZ
|
8.5 | Ki | 8 | Yes | |
QNOOVTZVMOOSAW
|
8.5 | IC50 | 4 | — | |
QNOOVTZVMOOSAW
|
8.5 | IC50 | 3 | — | |
SJHYJOUKZAHFOM
|
8.5 | IC50 | 3 | Yes | |
SYCRYYILCMOTOI
|
8.5 | IC50 | 3 | — | |
GTTSANJRVQIGFM
|
8.5 | IC50 | 3 | — | |
LPSBYKLLJOVSHM
|
8.5 | IC50 | 2 | — | |
WWOGYCVPNPHFGR
|
8.5 | IC50 | 2 | — | |
AUOYWLMHWSCDQP
|
8.5 | Ki | 2 | — | |
FQYLJBVSYHZWLT
|
8.5 | Ki | 35 | Yes | |
GSXRCPJTNIGKSZ
|
8.5 | Ki | 43 | — | |
LDGFTLHOBZCPLF
|
8.5 | Ki | 2 | — | |
MTCHQDWUHQADSY
|
8.5 | Ki | 29 | — | |
MVJMMLFMPWITEJ
|
8.5 | Ki | 110 | — | |
KAQWYRBKYUAJGJ
|
8.5 | IC50 | 2 | — | |
IMDKLXHGHQNHPQ
|
8.5 | IC50 | 2 | — | |
NXUFRHVUTNXZQT
|
8.5 | IC50 | 2 | — | |
OSOQQRUVRRWBMV
|
8.5 | IC50 | 3 | — | |
QHLGSHJIJSOCMR
|
8.5 | IC50 | 3 | — | |
QTBWCSQGBMPECM
|
8.5 | IC50 | 21 | Yes | |
WNQHVGYFQUHRNW
|
8.5 | Ki | 4 | — | |
FCZJOUALYCXWEB
|
8.5 | IC50 | 2 | — | |
GEQPKDUYCDTQRY
|
8.5 | IC50 | 2 | — | |
IDGLADROFDGGQO
|
8.5 | IC50 | 2 | — | |
VUEJUOUQJKHUSF
|
8.5 | IC50 | 2 | — | |
YRNDLUNPBSSFMF
|
8.5 | IC50 | 3 | — | |
ONTKIUFMGHVNJP
|
8.4 | IC50 | 3 | Yes | |
PJYYVACVVUDTRN
|
8.4 | IC50 | 3 | — | |
LAQKCNTWJTZLBG
|
8.4 | IC50 | 2 | — | |
MTPDPEHTPPGPLH
|
8.4 | IC50 | 3 | — | |
SXRUTBTWKQVBSM
|
8.4 | IC50 | 3 | — | |
VBXXGYSKTLTOBL
|
8.4 | IC50 | 2 | — | |
ACNCCUVYXQGPKZ
|
8.4 | Ki | 31 | — | |
ALKJNCZNEOTEMP
|
8.4 | Kd | 55 | — | |
BJLXYCDZTRNOAH
|
8.4 | IC50 | 3 | — | |
BRXHKUKMMZTVRE
|
8.4 | IC50 | 3 | — | |
CFIBXVQLBVNOHW
|
8.4 | Ki | 64 | — | |
GCBJDOWIQHMCMR
|
8.4 | Ki | 84 | — | |
GCYXEGSPUDSZJY
|
8.4 | Ki | 82 | — | |
GNSDDKAAHUFOKJ
|
8.4 | IC50 | 3 | — | |
GTZZCMNHEPBQEO
|
8.4 | IC50 | 2 | — | |
HCDXOVUMIOIELK
|
8.4 | IC50 | 3 | — | |
ITHCVKSAZKJITB
|
8.4 | IC50 | 2 | — | |
IVUGFMLRJOCGAS
|
8.4 | IC50 | 9 | — | |
JIKLDOKHOPBGQI
|
8.4 | IC50 | 3 | — | |
KLZCFIRMAFXIKI
|
8.4 | IC50 | 3 | — | |
KZDYTAXBOFTVGN
|
8.4 | IC50 | 3 | — | |
LLSACPYCBRAUIJ
|
8.4 | IC50 | 2 | — | |
LVECPYVAIBNSRV
|
8.4 | Ki | 33 | — |