Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JCZBWICLNFNCMR
|
6.0 | Ki | 9 | — | |
JOAWBRMGMMCJGS
|
6.0 | IC50 | 4 | Yes | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
LDHYCINFJPCBRY
|
6.0 | Ki | 9 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MASJMHFQMYAPJR
|
6.0 | Ki | 41 | — | |
MCKPYPWHBUXLEZ
|
6.0 | Ki | 21 | — | |
MGNQNQOSSLCUFP
|
6.0 | Ki | 12 | — | |
NEWAULHLLUCDPD
|
6.0 | Ki | 27 | — | |
OBHMNLIBIPFXCY
|
6.0 | Ki | 15 | — | |
ODNOTLMFNVWFTJ
|
6.0 | Ki | 11 | — | |
OETCTXGISYWYMV
|
6.0 | Ki | 7 | — | |
PAIFYAZSILXLBO
|
6.0 | Ki | 26 | — | |
PBCVBUZBZRHMQH
|
6.0 | Ki | 2 | — | |
PBNKREGCQAYWMQ
|
6.0 | Ki | 5 | — | |
PDBPUXLUVDSLML
|
6.0 | Ki | 14 | — | |
PVHJMAGWKQFOQA
|
6.0 | IC50 | 3 | — | |
RRNINKNJSOMCSD
|
6.0 | IC50 | 2 | — | |
RXVOXSGTUROJOL
|
6.0 | Ki | 11 | — | |
SBEXUUCHJQBRNW
|
6.0 | IC50 | 2 | — | |
SBWCIJOOABLPME
|
6.0 | Ki | 13 | — | |
TXXYVBLFLGPQOR
|
6.0 | IC50 | 5 | Yes | |
UTMRCMCLMBDPNW
|
6.0 | Ki | 10 | — | |
XTVULKIROSNNTG
|
6.0 | Ki | 29 | — | |
YDWMUCKJUNLURC
|
6.0 | Ki | 24 | — | |
YUOWJICKAJQZLS
|
6.0 | Ki | 35 | — | |
YXUQWISLOFXNGN
|
6.0 | Ki | 16 | — | |
ZLLCVOJWNDZXIO
|
6.0 | Ki | 11 | — | |
ZQVQTUFEKLITNT
|
6.0 | Ki | 10 | — |