Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AQKQATGZIKRZMQ
|
6.1 | Ki | 16 | — | |
DADQIQQXJSXLAV
|
6.1 | Ki | 5 | — | |
DJXMOVBYEXHLBK
|
6.1 | IC50 | 2 | — | |
DPYASQWYHILTBI
|
6.1 | IC50 | 6 | Yes | |
FATFDRYYCYZBQB
|
6.1 | IC50 | 5 | Yes | |
FDBPGAHVEGEARY
|
6.1 | Ki | 19 | — | |
GWJHMRBQEUHFOC
|
6.1 | Ki | 42 | — | |
HATNHAMXMKJCEI
|
6.1 | Ki | 9 | — | |
HFNKQEVNSGCOJV
|
6.1 | Ki | 18 | — | |
IMQVBCRZLIQNPG
|
6.1 | IC50 | 5 | Yes | |
JHVBIUJTSAGFKH
|
6.1 | IC50 | 2 | — | |
JPOSFPUHBHRUAX
|
6.1 | Ki | 40 | Yes | |
JRLSUZIPUYDUKX
|
6.1 | Ki | 22 | — | |
LJKJYKWDLJUZHA
|
6.1 | Ki | 24 | — | |
LZKFDPIUYGTKHZ
|
6.1 | IC50 | 3 | — | |
NXTQOFQOBODYSP
|
6.1 | IC50 | 2 | — | |
ODRSUVBAJITCIK
|
6.1 | IC50 | 2 | — | |
OEEGUWWPGAZRIJ
|
6.1 | Ki | 21 | — | |
PYWVRRARNRCHNK
|
6.1 | IC50 | 2 | — | |
QLWUDWMYFSWGHK
|
6.1 | Ki | 22 | — | |
QVNZKVACBBTKSL
|
6.1 | Ki | 38 | — | |
SDTHQOXRWZXTJF
|
6.1 | Ki | 16 | — | |
SHZPFCZPWGVEED
|
6.1 | Ki | 5 | — | |
SODGZPDNROVASD
|
6.1 | Ki | 7 | — | |
SVUIYNKSDCANAY
|
6.1 | Ki | 16 | — | |
TUDIKYFSCUIAIT
|
6.1 | Ki | 8 | — | |
USYYTOCVNAELEK
|
6.1 | IC50 | 3 | — | |
WFJYZRKNRWYRTN
|
6.1 | IC50 | 3 | — | |
XCOSAQGGGZDYJN
|
6.1 | IC50 | 11 | — | |
XUFLBSMTYMFOQH
|
6.1 | Ki | 43 | — | |
YKJSWMAVAKRUAN
|
6.1 | Ki | 19 | — | |
YNXZLNOLQBAZNQ
|
6.1 | IC50 | 3 | — | |
YOVNFNXUCOWYSG
|
6.1 | Ki | 33 | Yes | |
ZKZXNDJNWUTGDK
|
6.1 | Ki | 14 | — | |
CULJEMIZFZIMCZ
|
6.1 | Ki | 2 | — | |
DTHIPVGUOHBTJC
|
6.1 | IC50 | 2 | — | |
VHIUYJBYHQFWHD
|
6.1 | IC50 | 2 | — | |
WULUGQONDYDNKY
|
6.1 | IC50 | 5 | — | |
CTJAMSGCMYAVCZ
|
6.1 | Ki | 14 | — | |
DADQIKMIYWQYKT
|
6.1 | IC50 | 3 | — | |
DZLVIIVTIVFGQO
|
6.1 | IC50 | 2 | — | |
JFIZOYQARFPKTF
|
6.1 | IC50 | 2 | — | |
JJQRFOFBCUENFJ
|
6.1 | IC50 | 2 | — | |
RKFHHTFCUQMIGM
|
6.1 | IC50 | 3 | — | |
VMQANPBVERMFIJ
|
6.1 | IC50 | 2 | — | |
WWPZBBQLQAEXGE
|
6.1 | IC50 | 3 | — | |
ZBLXMVSBOPAZEE
|
6.1 | IC50 | 2 | — | |
DCQUEYKYABNNDA
|
6.1 | IC50 | 5 | Yes | |
HSVPJHAMWLJGAL
|
6.1 | IC50 | 2 | — | |
JYCUVOXSZBECAY
|
6.1 | IC50 | 6 | Yes |