Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FKBXSMMSZMPOPT
|
6.2 | IC50 | 2 | — | |
GPPDWFNQVHJOEU
|
6.2 | IC50 | 3 | — | |
HHJSKDRCUMVWKF
|
6.2 | IC50 | 7 | — | |
KJMALBRUCRDMTE
|
6.2 | IC50 | 6 | Yes | |
OSLOTHHIYWJTNJ
|
6.2 | IC50 | 3 | — | |
PBCZSGKMGDDXIJ
|
6.2 | Kd | 68 | Yes | |
PEPCSEJJADXCRB
|
6.2 | Ki | 4 | Yes | |
QCHJTTRZNFGGKY
|
6.2 | IC50 | 2 | — | |
ZLQITNSQCVUIPF
|
6.2 | IC50 | 2 | — | |
ZYYNXHSAMWEIKK
|
6.2 | IC50 | 4 | Yes | |
AFWWHBTVEBALQB
|
6.2 | IC50 | 2 | — | |
IDKYOQDTCCUVIN
|
6.2 | IC50 | 3 | — | |
LICZLVVAGKBEKQ
|
6.2 | IC50 | 3 | — | |
LIUOIZMHHPJCCK
|
6.2 | IC50 | 2 | — | |
LUPFUUDPZIMLMJ
|
6.2 | IC50 | 2 | — | |
USUYXDKUCNQBKM
|
6.2 | IC50 | 3 | — | |
WKBCIZTZDKGBEO
|
6.2 | IC50 | 3 | Yes | |
YZSOMODRJHNWOR
|
6.2 | IC50 | 3 | — | |
IAYGCINLNONXHY
|
6.2 | Kd | 50 | — | |
MNYJXBQMADDOQS
|
6.2 | IC50 | 3 | — | |
CKCGBVCGRTYHGB
|
6.1 | IC50 | 2 | — | |
JBZRAEUHDPMQSF
|
6.1 | IC50 | 34 | — | |
JVXJMEFHHQBIIG
|
6.1 | IC50 | 3 | Yes | |
JVXJMEFHHQBIIG
|
6.1 | IC50 | 2 | — | |
MLSFACRPOXXXGI
|
6.1 | IC50 | 2 | — | |
ZCGDFAQAYLXLJV
|
6.1 | IC50 | 2 | Yes | |
AAEYSRYWDWVNOK
|
6.1 | IC50 | 2 | — | |
GRIONNZJVZNNLU
|
6.1 | IC50 | 2 | — | |
IILGZBCIXYOQFH
|
6.1 | IC50 | 2 | — | |
MMUWRPSFAYHCTP
|
6.1 | IC50 | 3 | — | |
TWPZRFZCHZSVKG
|
6.1 | IC50 | 4 | — | |
TYJOLBATVWRDJW
|
6.1 | IC50 | 3 | — | |
VSDZCJADMNPBKB
|
6.1 | IC50 | 3 | — | |
YQQZZYYQTCPEAS
|
6.1 | IC50 | 2 | — | |
ZAYNEDGQOVESHF
|
6.1 | IC50 | 2 | — | |
GABKCBKPNYHAJC
|
6.1 | IC50 | 3 | — | |
IFTCXKUSJMWVRD
|
6.1 | IC50 | 7 | Yes | |
ISIXTEBAUAVHHA
|
6.1 | IC50 | 2 | — | |
NMULSNNATHYGPZ
|
6.1 | IC50 | 3 | Yes | |
OEYFMLOBJAFTAB
|
6.1 | IC50 | 3 | — | |
UXHHASKNWWRBLI
|
6.1 | IC50 | 3 | — | |
WROHCHCGJIWAPG
|
6.1 | IC50 | 3 | — | |
XVTGWJWSWNCTFK
|
6.1 | IC50 | 3 | — | |
DZERDSCGHZUEAK
|
6.1 | IC50 | 2 | — | |
GOYMLVLLBBEUKR
|
6.1 | IC50 | 2 | — | |
JODNFBDDCMSPPR
|
6.1 | IC50 | 2 | — | |
KSZAIPSQJXGBNH
|
6.1 | IC50 | 3 | — | |
UHRNXUUGHMAQNH
|
6.1 | IC50 | 2 | — | |
VPXPFQKSFBPCEO
|
6.1 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.1 | Ki | 50 | Yes |