Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVHDAKLRGJSVKQ
|
6.2 | IC50 | 4 | — | |
WAURSSMPBFMZPD
|
6.2 | IC50 | 2 | — | |
ZVFOBWUNGPKXSL
|
6.2 | IC50 | 3 | — | |
AEMIQVWOMZDMIJ
|
6.2 | IC50 | 3 | — | |
CWBWMDSAVFJNAD
|
6.2 | Ki | 7 | — | |
DZGATJHVQUFYSK
|
6.2 | Ki | 12 | — | |
FFFPNQJGIVIKKA
|
6.2 | Ki | 6 | — | |
FYRQDEVTRMEZHR
|
6.2 | Ki | 7 | — | |
GDYZFFBMSBDTAA
|
6.2 | Ki | 60 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
KMNQWCTYNHJINU
|
6.2 | IC50 | 2 | — | |
KSBWPNWWWVOGJM
|
6.2 | IC50 | 2 | — | |
MMNDBWXSYKZKAE
|
6.2 | IC50 | 5 | — | |
OLVBAUVSICCWEJ
|
6.2 | Ki | 39 | — | |
OWFLADWRSCINST
|
6.2 | Ki | 30 | — | |
PKCDDUHJAFVJJB
|
6.2 | Ki | 13 | — | |
RKUKAACYUCUJEE
|
6.2 | Ki | 58 | — | |
RZPPWTZTEBXBDQ
|
6.2 | IC50 | 2 | — | |
SUULIUKTZNKMMB
|
6.2 | Ki | 10 | — | |
UIRCQOKSJDLYBB
|
6.2 | Ki | 50 | — | |
UNVKXVCDLOLPJE
|
6.2 | Ki | 8 | — | |
VPCCZGPEHVCFOJ
|
6.2 | Ki | 2 | — | |
VUHNJTZMUNWJKN
|
6.2 | IC50 | 2 | — | |
VYPMKWZQENSPAB
|
6.2 | Ki | 3 | — | |
WINHZLLDWRZWRT
|
6.2 | Ki | 66 | — | |
WVGYXYZYFSSTFT
|
6.2 | IC50 | 2 | — | |
WWUXHXQJFWXACS
|
6.2 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
6.2 | IC50 | 8 | Yes | |
XNEPVLVYFUGJLF
|
6.2 | Ki | 27 | — | |
YWTBGJGMTBHQTM
|
6.2 | Ki | 65 | — | |
ZBYGBITZFKOQTA
|
6.2 | Ki | 18 | — | |
CYXVEZJWVJIFPJ
|
6.2 | IC50 | 4 | Yes | |
DUKJABPGWUISRC
|
6.2 | IC50 | 3 | — | |
GSYZCTCPLRSRGI
|
6.2 | IC50 | 2 | — | |
HCCIPHZGDVGCQS
|
6.2 | IC50 | 2 | — | |
HLVQIKPORSSRAI
|
6.2 | IC50 | 3 | — | |
HWXVIOGONBBTBY
|
6.2 | Kd | 27 | — | |
IOBDCMVQCAWFQQ
|
6.2 | IC50 | 2 | — | |
JGWRKYUXBBNENE
|
6.2 | IC50 | 11 | — | |
OEWIUKZNWRWPFA
|
6.2 | IC50 | 3 | — | |
FJKSYFWQWKRPJT
|
6.2 | IC50 | 2 | — | |
FRJOVFNLSNXELB
|
6.2 | IC50 | 3 | — | |
MZOWKBSAYUJCKQ
|
6.2 | IC50 | 2 | — | |
OHDDAHALDZFALJ
|
6.2 | IC50 | 3 | — | |
RYGAYBGVUQJRJA
|
6.2 | IC50 | 3 | — | |
ULDURKNHYFYKMS
|
6.2 | IC50 | 3 | — | |
XKZQZMSAWVDRSP
|
6.2 | IC50 | 39 | Yes | |
AMKGWZMBMZFCTO
|
6.2 | IC50 | 3 | — | |
CMLSWGVOCIGIAK
|
6.2 | IC50 | 2 | — | |
DIOOREPVPOCQKL
|
6.2 | IC50 | 4 | Yes |