Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
JXPRLYUMECVOOZ
|
6.3 | IC50 | 2 | — | |
KTUZOTUSWXJDIS
|
6.3 | IC50 | 3 | — | |
LJPXHKWPVWLKRN
|
6.3 | IC50 | 3 | — | |
LLROFEFDEFKWQN
|
6.3 | IC50 | 3 | — | |
MCXNJEWRZUGGHR
|
6.3 | Ki | 5 | Yes | |
SWQVIBOZAHRMDS
|
6.3 | IC50 | 2 | — | |
VTMZVLJPBOBMNY
|
6.3 | IC50 | 2 | — | |
AEYLJTAIDDIOBA
|
6.3 | Ki | 53 | — | |
BDDMFFMPRZTZGH
|
6.3 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
6.3 | Ki | 60 | — | |
BXSXPCFESWIUHR
|
6.3 | IC50 | 3 | — | |
CQXFMKMVOOUGSS
|
6.3 | Ki | 6 | — | |
DBKQWGCVGCVPIP
|
6.3 | Ki | 21 | — | |
DFMCXVONDDGQIY
|
6.3 | Ki | 66 | — | |
DPEXRCOBPACFOO
|
6.3 | Ki | 36 | — | |
FUMCKNCUEAQHCV
|
6.3 | Ki | 103 | — | |
GDOTWXUDXHZXHG
|
6.3 | Ki | 3 | — | |
HDRLAVNNWSHSOA
|
6.3 | Ki | 19 | — | |
HSKVRPZJBMXFDX
|
6.3 | Ki | 20 | — | |
IJRBJCMLWLFMIN
|
6.3 | Ki | 17 | — | |
KSBCGWKXTJXPLL
|
6.3 | IC50 | 3 | — | |
MDZNNHJKFFMBHO
|
6.3 | IC50 | 2 | — | |
MIYRKQLKDQNUKZ
|
6.3 | Ki | 23 | — | |
OQNPAZRZCXFOBC
|
6.3 | Ki | 11 | — | |
PNAPQQCRNHMIER
|
6.3 | Ki | 12 | — | |
QAPDXRHCCUUBNB
|
6.3 | IC50 | 2 | — | |
RHIXHHWKASAAHP
|
6.3 | IC50 | 2 | — | |
RIBBPSYZBQQTQC
|
6.3 | Ki | 15 | — | |
SWQVIBOZAHRMDS
|
6.3 | IC50 | 3 | Yes | |
UEIRKXUBXCSHJE
|
6.3 | Ki | 19 | — | |
UVBKNBPCVRBUTF
|
6.3 | IC50 | 5 | — | |
WCRYRBRNFCXTTR
|
6.3 | IC50 | 4 | Yes | |
WOTLXQZLXOXMFD
|
6.3 | Ki | 7 | — | |
WUBHCQHBUVGGRX
|
6.3 | Ki | 11 | — | |
XBDWKVLCDCUNHH
|
6.3 | Ki | 18 | — | |
XEGSWNKCRGYRFG
|
6.3 | IC50 | 3 | — | |
XSXNOQJYDZWMGX
|
6.3 | IC50 | 2 | — | |
XZWVOUQIYLZUCJ
|
6.3 | Ki | 23 | — | |
DWCZEZXJZXJTHE
|
6.3 | IC50 | 6 | Yes | |
LEFKZSWCBZBDLU
|
6.3 | IC50 | 5 | Yes | |
PBBRUKZHVDWECM
|
6.3 | IC50 | 3 | — | |
RKGNVOKYSGKVQZ
|
6.3 | IC50 | 7 | Yes | |
YLKJJERCKRGNPB
|
6.3 | IC50 | 2 | Yes | |
ZOAKQENCPNJUTG
|
6.3 | IC50 | 2 | — | |
ALGXUTHRGCWFHE
|
6.3 | IC50 | 2 | — | |
CAQMYVREIKAKFV
|
6.3 | IC50 | 2 | — | |
RIBFZRWGJCKRQH
|
6.3 | IC50 | 3 | Yes | |
TZKMWKXQVXWVFE
|
6.3 | IC50 | 2 | — | |
UJLAWZDWDVHWOW
|
6.3 | Kd | 16 | — |