Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DHGCUTOPNQKCLE
|
6.4 | IC50 | 2 | — | |
DZSFRHLIEUXICV
|
6.4 | IC50 | 2 | — | |
GJFMMVDSDLIPNN
|
6.4 | IC50 | 2 | — | |
GVWOZWUDWKTPQX
|
6.4 | IC50 | 2 | — | |
HJDDOMBYBZNDRI
|
6.4 | IC50 | 2 | — | |
JHIXLFUYHWBARZ
|
6.4 | IC50 | 2 | — | |
OJEKLDYMEMWETM
|
6.4 | IC50 | 2 | — | |
UTCDALCXQDRSJR
|
6.4 | IC50 | 2 | — | |
XMKPDQSYIWBQMS
|
6.4 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
CERFFPJDBQMQTN
|
6.4 | IC50 | 2 | — | |
CXKZYGHFQYYGMN
|
6.4 | IC50 | 2 | — | |
DVCNPIFFEMVJNY
|
6.4 | IC50 | 3 | — | |
GWTSGLRTAKOPSF
|
6.4 | IC50 | 3 | — | |
PZVIQPBSJBPATG
|
6.4 | IC50 | 2 | Yes | |
LKZXAQZZOSZHLE
|
6.4 | IC50 | 3 | — | |
MEKHYJNJENZTPN
|
6.4 | IC50 | 3 | Yes | |
MEKHYJNJENZTPN
|
6.4 | IC50 | 2 | — | |
MLDQJTXFUGDVEO
|
6.4 | Kd | 85 | Yes | |
PSRQKGSEEYKFMK
|
6.4 | IC50 | 2 | — | |
QQOUQSHLYUUNAH
|
6.4 | IC50 | 2 | — | |
REXOPODAAFIDIW
|
6.4 | IC50 | 2 | — | |
SSHDKAJDJAVHAF
|
6.4 | IC50 | 8 | Yes | |
USSPDYYDWFNICI
|
6.4 | IC50 | 2 | Yes | |
VGBYAYCYPVFDTM
|
6.4 | IC50 | 6 | — | |
WDDYOKLMIHMUSU
|
6.4 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
6.4 | Kd | 46 | — | |
CBAXBOKSVQWPAQ
|
6.3 | IC50 | 2 | — | |
CEONSWRDFKMFNM
|
6.3 | IC50 | 2 | — | |
KGJQVQSYWYQQOD
|
6.3 | IC50 | 2 | — | |
MTIWAQLYXOZHBE
|
6.3 | IC50 | 2 | — | |
NQFJXYKOQSRMCX
|
6.3 | Ki | 4 | Yes | |
USCOCXHLSIVHKU
|
6.3 | IC50 | 3 | — | |
BIGXOFQDFCWJGU
|
6.3 | IC50 | 3 | — | |
FQIKRDSTMHHCGU
|
6.3 | IC50 | 3 | — | |
IOZKFIAWEQJPPC
|
6.3 | IC50 | 2 | — | |
NQLBAFDUCAUTMR
|
6.3 | IC50 | 2 | — | |
OLDWHOFNZYPPSR
|
6.3 | IC50 | 2 | — | |
PIHRITDRJRTFQR
|
6.3 | IC50 | 2 | — | |
QHQWGJPISLNJMT
|
6.3 | IC50 | 3 | Yes | |
TYTPWTMXQPOHQI
|
6.3 | IC50 | 2 | — | |
VMUFFHDFTBDUIP
|
6.3 | IC50 | 2 | — | |
VNDDOAWIHYNTOI
|
6.3 | IC50 | 3 | — | |
AFPQNJFINOFINI
|
6.3 | IC50 | 3 | — | |
FOJFMSKCYTZGMD
|
6.3 | IC50 | 3 | — | |
IBWUYNSLISMPFY
|
6.3 | IC50 | 4 | — | |
IUDBEIQBJIEKNX
|
6.3 | IC50 | 3 | — | |
JAHXQCZCZURPTI
|
6.3 | IC50 | 34 | — | |
QBIUCEGPYOMVEE
|
6.3 | IC50 | 3 | — | |
GMYYMEOGFRKSFS
|
6.3 | IC50 | 29 | — |