Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RWFVTYXPQZEJCN
|
6.4 | IC50 | 3 | — | |
BQOUQYBZXHHCIK
|
6.4 | IC50 | 2 | — | |
FNLDEFMOSGPZBB
|
6.4 | IC50 | 3 | — | |
LYTYIKFSJLZITL
|
6.4 | IC50 | 2 | — | |
PGINJTUIQUFAPP
|
6.4 | IC50 | 4 | Yes | |
VXWLORZXKCHFJR
|
6.4 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
AMOJCASSAZNSPN
|
6.4 | IC50 | 3 | — | |
DBLHAVCJDSOAAZ
|
6.4 | IC50 | 2 | — | |
DLHDVXKHPFNZCD
|
6.4 | IC50 | 2 | — | |
GBLWEKVVBOPDQK
|
6.4 | IC50 | 2 | — | |
HSAQBRJGYZIVJP
|
6.4 | IC50 | 5 | Yes | |
MPVGZUGXCQEXTM
|
6.4 | Kd | 61 | Yes | |
UXCOLBRRXSIGNA
|
6.4 | IC50 | 2 | — | |
VUYHYBMHVWMAIB
|
6.4 | IC50 | 2 | — | |
XZXDFCJIGPPSNH
|
6.4 | IC50 | 2 | — | |
YCZYGQPCRPOGLT
|
6.4 | IC50 | 3 | — | |
YGKBBMAZIAXASO
|
6.4 | IC50 | 3 | — | |
BNLPAUPVSCPTDM
|
6.4 | Ki | 15 | — | |
CLAFAHXMXSENJP
|
6.4 | Ki | 3 | — | |
COWZMOOYUJTEOM
|
6.4 | IC50 | 2 | — | |
DPRNXTSMYVCYLJ
|
6.4 | IC50 | 13 | — | |
FDVSOQRNTAPCHB
|
6.4 | Ki | 40 | — | |
FONINLXADYUZFI
|
6.4 | Ki | 25 | — | |
FRAYTYRDTFKQRS
|
6.4 | IC50 | 2 | — | |
FZMCQVGUQKFBIJ
|
6.4 | IC50 | 4 | — | |
HVNQYDHDQBJAAH
|
6.4 | IC50 | 3 | Yes | |
KIUHBHFVVQQALF
|
6.4 | Ki | 9 | — | |
MTOXIGVDKCMGPO
|
6.4 | IC50 | 2 | — | |
NGQVGKKCRFIRQR
|
6.4 | IC50 | 3 | — | |
NLDZIKOJZCTRAZ
|
6.4 | Ki | 5 | — | |
OIDZQWOKVFYZSD
|
6.4 | Ki | 8 | — | |
OQSVYNYDHYYKJX
|
6.4 | Ki | 7 | — | |
OWDRQHVEJIYVOI
|
6.4 | Ki | 47 | — | |
SJLQDZDKTVBBLP
|
6.4 | Ki | 9 | — | |
TXHOCWWJSGCZLC
|
6.4 | Ki | 18 | — | |
VSVKFEMFAYXZKR
|
6.4 | Ki | 14 | Yes | |
VXYDJXMHISGSDA
|
6.4 | Ki | 59 | — | |
WYLTWMHCCIFULE
|
6.4 | IC50 | 2 | — | |
WYLTWMHCCIFULE
|
6.4 | IC50 | 3 | Yes | |
XJKZZPPHNXWMOR
|
6.4 | IC50 | 2 | — | |
YEPNVBNYCRGZRX
|
6.4 | Ki | 26 | — | |
ZDXVFTIWQLMEIZ
|
6.4 | IC50 | 3 | — | |
CNMLMSRMIXOQJZ
|
6.4 | IC50 | 2 | — | |
IPIWNOAWKGRYOY
|
6.4 | IC50 | 4 | Yes | |
MOVPUGMNBIXRIN
|
6.4 | IC50 | 2 | — | |
QOYWSCMDSDPETI
|
6.4 | IC50 | 2 | — | |
SIXVRXARNAVBTC
|
6.4 | IC50 | 12 | — | |
VOJAEHGONMEHQB
|
6.4 | IC50 | 2 | — | |
CPSQBCZJMZEPOE
|
6.4 | IC50 | 2 | Yes |