Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLLDNGSQDXHYQI
|
6.5 | IC50 | 2 | — | |
PUPCRRRSBUYJAD
|
6.5 | Ki | 44 | Yes | |
QYAOLXACVZFCGN
|
6.5 | IC50 | 2 | — | |
SBFPHSVZEXSHTL
|
6.5 | Ki | 62 | — | |
UGKORVWYIOIXIN
|
6.5 | IC50 | 2 | — | |
VRIFJAKXSBXYFZ
|
6.5 | Ki | 8 | — | |
XFWUTMHVDGPWLH
|
6.5 | Ki | 75 | — | |
XUGXUDSTKPTWNB
|
6.5 | Ki | 10 | — | |
XZTYFGBEDWNFPM
|
6.5 | IC50 | 3 | — | |
YKYRQCWLYUTVIE
|
6.5 | Ki | 16 | — | |
YNVBUFWEFFQVHM
|
6.5 | Ki | 3 | — | |
YUNGWKDFWCZWAM
|
6.5 | IC50 | 2 | — | |
CEUGFEWLHGCQEO
|
6.5 | IC50 | 2 | — | |
GYMQBVYIGPAFNJ
|
6.5 | IC50 | 2 | — | |
LVJOSXIHDWKFCU
|
6.5 | IC50 | 3 | — | |
OFJINLPIXOGONH
|
6.5 | IC50 | 2 | — | |
WKWGFJFNCXAUEX
|
6.5 | Ki | 14 | Yes | |
AKPRVQKEQOLLND
|
6.5 | IC50 | 3 | — | |
CBRMHVZZHXKJJW
|
6.5 | IC50 | 2 | — | |
JIJFEPIYIIFIDK
|
6.5 | IC50 | 3 | — | |
LSOJMWRTJMDWFW
|
6.5 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
6.5 | Kd | 151 | — | |
CULXCGPBYYEBGM
|
6.5 | IC50 | 2 | Yes | |
DTEKTGDVSARYDS
|
6.5 | IC50 | 11 | — | |
GIBXNJNDDSOAHX
|
6.5 | IC50 | 2 | — | |
HAYYBYPASCDWEQ
|
6.5 | IC50 | 47 | — | |
HUKDVVBUBJTWCJ
|
6.5 | IC50 | 2 | — | |
KXEVSPQLDCBMPG
|
6.5 | IC50 | 2 | — | |
YJPSFRIIFNZTAR
|
6.5 | IC50 | 2 | — | |
HFEPCQCRRRINGD
|
6.5 | IC50 | 2 | — | |
MVKSHUDBXVAUPP
|
6.5 | IC50 | 2 | — | |
RPMDNLSTGYONBC
|
6.5 | IC50 | 3 | — | |
BZDPNSHFCIPOPU
|
6.5 | IC50 | 2 | Yes | |
HOZCGFJBIZZKTL
|
6.5 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
6.5 | Kd | 88 | Yes | |
LBJUQENGWONWHC
|
6.5 | IC50 | 2 | — | |
MOAAJQGICJEPNH
|
6.5 | IC50 | 2 | — | |
VVFYYEUTPUGPNR
|
6.5 | IC50 | 2 | — | |
WTCMEZGTRYAQQE
|
6.5 | IC50 | 3 | — | |
IHHQKCHZXRIDLL
|
6.4 | IC50 | 2 | — | |
JLBAXNKYJZOYGQ
|
6.4 | IC50 | 4 | Yes | |
NNCYMIKCSDIHJR
|
6.4 | IC50 | 3 | — | |
ONWUZLTWJSDCTN
|
6.4 | IC50 | 2 | — | |
PIAOPVOJTUSVEB
|
6.4 | IC50 | 3 | — | |
PMDUMOUXISSZED
|
6.4 | IC50 | 3 | — | |
ZORWXMUNOJMUBY
|
6.4 | IC50 | 2 | — | |
ZRBJCFDMMPLPCO
|
6.4 | IC50 | 2 | — | |
DQPVIVGCZVQZDO
|
6.4 | IC50 | 3 | — | |
KYEHLWMHQXZVMF
|
6.4 | IC50 | 2 | — | |
MBNSFOGJHWUIOY
|
6.4 | IC50 | 2 | — |