Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DNGHYRYQEMRIDG
|
6.5 | IC50 | 3 | — | |
LSVRKVVHCSGSCC
|
6.5 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.5 | Kd | 137 | Yes | |
BLQYVHBZHAISJM
|
6.5 | IC50 | 21 | Yes | |
HMYRVBUHXWGRJY
|
6.5 | IC50 | 2 | — | |
JQBQAGHSJMBPSH
|
6.5 | IC50 | 6 | — | |
NROKZPYRSOKBHT
|
6.5 | IC50 | 3 | Yes | |
RSIMWZIJZCXPJV
|
6.5 | IC50 | 3 | Yes | |
WUTLVPJTLNYGRZ
|
6.5 | IC50 | 2 | — | |
YKPYZRLLGKAMJE
|
6.5 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
6.5 | IC50 | 54 | — | |
JXJVDYZUMYOTJW
|
6.5 | IC50 | 3 | — | |
KVBBSBPIPKLJCO
|
6.5 | IC50 | 3 | — | |
NROKZPYRSOKBHT
|
6.5 | IC50 | 2 | — | |
RIZUAVMTLJDZPO
|
6.5 | IC50 | 2 | — | |
FNZJYDYAQSDVIG
|
6.5 | IC50 | 2 | — | |
LLHGFGUOUWJTLQ
|
6.5 | IC50 | 3 | — | |
NYMXQEKCEGCXNT
|
6.5 | IC50 | 3 | Yes | |
UJBJAMOSBBJZBK
|
6.5 | IC50 | 6 | Yes | |
XTULNCWAJUYUIA
|
6.5 | IC50 | 4 | — | |
AJHBYQLGRIOMIW
|
6.5 | IC50 | 3 | — | |
FFBJZTQMALZDTE
|
6.5 | IC50 | 2 | — | |
FHRXTSQACPDPRQ
|
6.5 | IC50 | 2 | Yes | |
GFDMYTNCMHUIAT
|
6.5 | IC50 | 2 | Yes | |
IDMDQNLKWPITHX
|
6.5 | IC50 | 3 | — | |
WHFRCTYFOGGZAU
|
6.5 | IC50 | 2 | Yes | |
XUGCPDXHIQDAKV
|
6.5 | IC50 | 2 | — | |
AARZYPZTMIRNPN
|
6.5 | Ki | 3 | — | |
AQZIXHSRFOGYHF
|
6.5 | Ki | 9 | — | |
BKBCSMDCCAWWNC
|
6.5 | Ki | 7 | — | |
BYMPQGHXDOZTHZ
|
6.5 | IC50 | 2 | — | |
CEUGFEWLHGCQEO
|
6.5 | IC50 | 3 | Yes | |
CFSAUVVSNYZBGZ
|
6.5 | IC50 | 2 | — | |
CTWASZOPAJRLED
|
6.5 | IC50 | 2 | — | |
CVWXJKQAOSCOAB
|
6.5 | Kd | 35 | — | |
FJZXDUKUMALHNP
|
6.5 | Ki | 10 | — | |
FPQHXFMYXQZPSV
|
6.5 | Ki | 23 | — | |
FPWMHTSISQKIJN
|
6.5 | IC50 | 2 | — | |
GEGCXGMFUYJULA
|
6.5 | Ki | 30 | Yes | |
HVNQYDHDQBJAAH
|
6.5 | IC50 | 3 | Yes | |
IBPSHHSPUPWXHN
|
6.5 | Ki | 6 | — | |
IUEBPIPDFMCSTP
|
6.5 | Ki | 29 | — | |
JTGMDPHLGBACAV
|
6.5 | IC50 | 5 | Yes | |
LCHCMNPPJLRNHX
|
6.5 | Ki | 3 | — | |
MMMPFWNSQKXKDX
|
6.5 | Ki | 14 | — | |
NMHMCXTYPRADBA
|
6.5 | Ki | 20 | — | |
OUJZYQBEFNDJQN
|
6.5 | Ki | 71 | — | |
PCQMERRARZKTPW
|
6.5 | Ki | 68 | — | |
PEXKNSGOEOREKM
|
6.5 | Ki | 13 | — | |
PJSBFZAYJQMORO
|
6.5 | Ki | 11 | — |