Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GSYNTOXSBKQRAW
|
6.6 | Ki | 7 | — | |
IIIJQZOSLLAVTL
|
6.6 | Ki | 2 | — | |
IVIGCDKRIYEDPR
|
6.6 | IC50 | 3 | Yes | |
JWQOJVOKBAAAAR
|
6.6 | Ki | 29 | — | |
LNIDFQVRZCDVBI
|
6.6 | Ki | 16 | — | |
LRDIEHDJWYRVPT
|
6.6 | Ki | 2 | — | |
NKGLJTITEFZKAN
|
6.6 | Ki | 35 | — | |
POSCFQVOEFKTSG
|
6.6 | IC50 | 3 | — | |
QBKUOOQFSVMDPB
|
6.6 | Ki | 31 | — | |
QNUKRWAIZMBVCU
|
6.6 | Ki | 46 | — | |
RWUJEVMUBYCUBS
|
6.6 | Ki | 3 | — | |
SGZZQKMOFHIDKW
|
6.6 | IC50 | 13 | — | |
STFRNQJMPQIRPD
|
6.6 | Ki | 2 | — | |
UGHBIMSDMGHFIE
|
6.6 | Ki | 10 | — | |
UTFXYGYVDDLJER
|
6.6 | Ki | 36 | — | |
VAKWGLDYQAWDPS
|
6.6 | Ki | 3 | Yes | |
VBNPWXWJZJNXEY
|
6.6 | Ki | 18 | Yes | |
WDARYLSSWBWVCU
|
6.6 | Ki | 49 | — | |
XAHJIRNRDAKTEF
|
6.6 | Ki | 18 | — | |
XIOOJUQFJYPVLA
|
6.6 | Ki | 17 | — | |
YEKVTSRZMPLPFK
|
6.6 | Ki | 17 | — | |
YFVHXPJXPIIXGA
|
6.6 | IC50 | 2 | — | |
ZGDYBJXDIXVTLV
|
6.6 | Ki | 54 | — | |
ZRQXCQXWTLVASO
|
6.6 | Ki | 36 | — | |
ZRTDSOVGBJZNBQ
|
6.6 | Ki | 3 | — | |
BNCUORANSSPIJN
|
6.6 | IC50 | 2 | — | |
CRIUUFBOLAJGNR
|
6.6 | IC50 | 3 | — | |
ABPYUTLLWASPRF
|
6.6 | IC50 | 2 | — | |
AOMMHIPSMLPJKQ
|
6.6 | IC50 | 4 | — | |
BVSXEPUYNGJRDW
|
6.6 | IC50 | 2 | — | |
DVKYBHNNFVMHIN
|
6.6 | IC50 | 3 | Yes | |
MZWALFBOTNMRTP
|
6.6 | IC50 | 7 | Yes | |
NSVICOOGAFNGHP
|
6.6 | IC50 | 2 | — | |
PNSDQTZGJZEYEU
|
6.6 | IC50 | 2 | — | |
VBAJQFDWESLMDW
|
6.6 | IC50 | 3 | — | |
YKVSMJHGYWIRDE
|
6.6 | IC50 | 2 | — | |
YZOZEZFNWLULHX
|
6.6 | IC50 | 2 | — | |
FLYNZEXUURBXAW
|
6.6 | IC50 | 6 | Yes | |
GBMDFZRFAMTRLI
|
6.6 | IC50 | 2 | — | |
HHCSNTXVZDWIGT
|
6.6 | IC50 | 2 | — | |
NALGZACUGTTXDW
|
6.6 | IC50 | 3 | — | |
PRASIGARSOSUQT
|
6.6 | IC50 | 11 | Yes | |
WEOGGUARIACEDQ
|
6.6 | IC50 | 2 | — | |
XXSQNJQHHHVCBG
|
6.6 | IC50 | 7 | Yes | |
YUPOZANDWNEEJQ
|
6.6 | IC50 | 3 | Yes | |
CZXWODTUMHNHMA
|
6.6 | IC50 | 2 | — | |
DQJRSRINKOLTGU
|
6.6 | IC50 | 2 | Yes | |
MXUDIOKQCGEJOI
|
6.6 | IC50 | 3 | — | |
UPVLUCLFYXJYAO
|
6.6 | IC50 | 2 | — | |
WKBADCPZJIWSRC
|
6.6 | IC50 | 2 | — |