Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GHXCSPGXRVESNT
|
9.0 | IC50 | 2 | — | |
GZEGBHAXGLPTQY
|
9.0 | IC50 | 2 | — | |
HOHHMYNNRAVKQB
|
9.0 | IC50 | 3 | Yes | |
JYUQCOURFHGOMR
|
9.0 | IC50 | 2 | — | |
KALSMXLQRKFVPO
|
9.0 | Ki | 3 | Yes | |
KSAUSYLGKMZHPT
|
9.0 | Ki | 3 | Yes | |
LNXKRNKFQNYAGZ
|
9.0 | Ki | 2 | — | |
LYDTZBUSUCDSRL
|
9.0 | IC50 | 3 | Yes | |
MRVCHPICZWIIEF
|
9.0 | IC50 | 3 | Yes | |
NMKNRNXEPYFWSY
|
9.0 | IC50 | 3 | — | |
NNQPYKAOGXIZBP
|
9.0 | IC50 | 2 | — | |
OBNJJMRMHFJKPW
|
9.0 | IC50 | 2 | — | |
PJXUDKNHESNHGD
|
9.0 | IC50 | 2 | — | |
SQYOZDZCDXQDRZ
|
9.0 | Ki | 3 | Yes | |
SVXYIHAHZMQVBU
|
9.0 | IC50 | 2 | — | |
VMAMZHADUWRQFW
|
9.0 | IC50 | 3 | — | |
WPASUZBJIGBQSX
|
9.0 | IC50 | 2 | — | |
WPDWJWPDAWEUDW
|
9.0 | IC50 | 3 | — | |
XHORJSJFHVABEA
|
9.0 | IC50 | 5 | — | |
XMSFPGDGANKHJW
|
9.0 | IC50 | 2 | — | |
ZQCJERNZTUANGM
|
9.0 | IC50 | 3 | — | |
CYGJLKBTKVKZQE
|
9.0 | IC50 | 6 | — | |
RQMCICOFYAOUFP
|
9.0 | IC50 | 2 | — | |
SHHVFBHRTMUGBM
|
9.0 | IC50 | 3 | — | |
SHTJDUVIHHPLRU
|
9.0 | IC50 | 2 | — | |
SKTCDUXPKLCJIP
|
9.0 | IC50 | 3 | — | |
SPWUNHDCOAYNOQ
|
9.0 | IC50 | 2 | — | |
DDSBMKNXVLTBPK
|
8.9 | IC50 | 3 | — | |
JGTLCWBXBNQZGX
|
8.9 | IC50 | 3 | — | |
PWWRGGQDPGYVDM
|
8.9 | IC50 | 3 | — | |
RCBPCGVUXHCRAA
|
8.9 | IC50 | 2 | — | |
VMAAFUOXTWPYRN
|
8.9 | IC50 | 9 | Yes | |
XTXMJKTXFRAXRP
|
8.9 | IC50 | 2 | — | |
YXUPBHOIGGKRNR
|
8.9 | IC50 | 2 | — | |
KMSYJPDFKRHHNJ
|
8.9 | Ki | 2 | — | |
ROIWTEBVYRJZEG
|
8.9 | Ki | 3 | — | |
CIDVBRKDJFCKQF
|
8.9 | IC50 | 2 | — | |
SRJJNRIRROSSLD
|
8.9 | IC50 | 3 | — | |
ZKQGSMFEXARYCS
|
8.9 | IC50 | 3 | — | |
PDULEZONFAQVLI
|
8.8 | IC50 | 3 | — | |
RGLSQZGEAOHRTM
|
8.8 | IC50 | 3 | — | |
UFMCGKYLIYMLOY
|
8.8 | IC50 | 3 | — | |
VTKXOUFYFLRSDX
|
8.8 | IC50 | 3 | Yes | |
VWYGEDAFWDXUMQ
|
8.8 | IC50 | 3 | — | |
BGVHRAAMOSNTDT
|
8.8 | IC50 | 2 | — | |
DHBOCWJFJJEPCN
|
8.8 | IC50 | 3 | Yes | |
JRUFBZGMCKTNQR
|
8.8 | IC50 | 5 | — | |
KCAURAAIHCEWSW
|
8.8 | IC50 | 3 | — | |
OIDHYGPWCABWGM
|
8.8 | IC50 | 3 | — | |
QSWPJTLRYDNNBP
|
8.8 | IC50 | 3 | — |