Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQIDEXUPWOIQDI
|
6.7 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
6.7 | IC50 | 47 | — | |
BGNRYQCGVJJPRI
|
6.7 | Ki | 3 | Yes | |
GBUDRABUNBYJKG
|
6.7 | IC50 | 7 | — | |
HXHAJRMTJXHJJZ
|
6.7 | IC50 | 52 | Yes | |
WOMKQOXPOGODKV
|
6.7 | IC50 | 3 | — | |
BBTDOQATPTVBOJ
|
6.7 | IC50 | 3 | Yes | |
BBTDOQATPTVBOJ
|
6.7 | IC50 | 2 | — | |
WQLHTTLATAQIEQ
|
6.7 | IC50 | 2 | — | |
ASOKHEVFZLQTPE
|
6.7 | Ki | 3 | Yes | |
FNVQWFPDIYQCSF
|
6.7 | IC50 | 8 | Yes | |
GDSIRLSWDHCACM
|
6.7 | IC50 | 2 | — | |
GJDYHJPLCHRKEK
|
6.7 | IC50 | 3 | — | |
HCLRALZLPGWRQY
|
6.7 | IC50 | 2 | — | |
KWZCYJXUMYBAAS
|
6.7 | IC50 | 2 | Yes | |
QSKHBRBUJVMKMR
|
6.7 | IC50 | 2 | — | |
UCKMYULEGLLJLE
|
6.7 | IC50 | 3 | Yes | |
GADYBZMYJCZJLX
|
6.7 | IC50 | 2 | — | |
ORYMWWSJZRCUSV
|
6.7 | IC50 | 7 | — | |
ZVIBNYVMRHMJFS
|
6.7 | IC50 | 3 | — | |
CHAZIKNZOXHZJA
|
6.6 | IC50 | 3 | — | |
JSKOFTDOVDUJQY
|
6.6 | IC50 | 2 | — | |
MFHCYEYXDLMXRP
|
6.6 | IC50 | 2 | — | |
NESZTHUOBRFWLA
|
6.6 | IC50 | 2 | — | |
XUAORJVHYWCADO
|
6.6 | Ki | 5 | Yes | |
ZCHJWXKREFTWSX
|
6.6 | IC50 | 2 | — | |
CBBZXHUFHIEZHP
|
6.6 | IC50 | 4 | — | |
CQJVDJZHNQFAOH
|
6.6 | IC50 | 2 | — | |
DKDRRZIRAAABEN
|
6.6 | IC50 | 2 | — | |
HWDCMQBNOROFEQ
|
6.6 | IC50 | 2 | — | |
JNAHXDJEKAMVMC
|
6.6 | IC50 | 3 | — | |
NTYYMMATFKHAFI
|
6.6 | IC50 | 2 | — | |
QLQCSGMKEZSDOV
|
6.6 | IC50 | 2 | — | |
TVLISAFENSCERO
|
6.6 | IC50 | 2 | — | |
UEMHNDHVZSSWDQ
|
6.6 | IC50 | 2 | — | |
VMUAYDSPKYLLJV
|
6.6 | IC50 | 3 | Yes | |
XCDJZSMEKBJHEE
|
6.6 | IC50 | 2 | — | |
XZDKAVSSXNBWNJ
|
6.6 | IC50 | 5 | Yes | |
HFPZHQLESGVWLH
|
6.6 | Kd | 2 | — | |
JDWRBLXGJZCOBR
|
6.6 | IC50 | 2 | — | |
PDOXJVQIOMGRBV
|
6.6 | IC50 | 2 | — | |
YPLADSZZPCZLET
|
6.6 | Ki | 3 | — | |
AYXVSCVVQIADBF
|
6.6 | Ki | 10 | — | |
CHTMRWQLNNRRFJ
|
6.6 | Ki | 70 | — | |
CLKZDZYGBHNPSM
|
6.6 | IC50 | 2 | — | |
FGVBXWYMYMNXGE
|
6.6 | IC50 | 4 | Yes | |
FPEIJQLXFHKLJV
|
6.6 | IC50 | 2 | — | |
FXKGUMKUGJEBFI
|
6.6 | IC50 | 2 | — | |
GASPHORHXIOCBB
|
6.6 | IC50 | 4 | Yes | |
GLDSKRNGVVYJAB
|
6.6 | IC50 | 16 | — |