Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BYWLEEWVFXOXAG
|
6.7 | IC50 | 2 | — | |
FVYYEKOHBWXBII
|
6.7 | IC50 | 2 | — | |
IABSWKZENVKESR
|
6.7 | IC50 | 3 | — | |
IIDXPMBKJWZQEU
|
6.7 | IC50 | 2 | — | |
JZMGYGRZHAFRMN
|
6.7 | IC50 | 2 | Yes | |
LROSTRBOAUSAAK
|
6.7 | IC50 | 2 | — | |
REKQXOMQYIHNKM
|
6.7 | IC50 | 3 | Yes | |
VTYQURZUYOUAOK
|
6.7 | IC50 | 3 | — | |
YLDZSOOIPBFXEN
|
6.7 | IC50 | 3 | — | |
YOFJPZPGHXWQJB
|
6.7 | IC50 | 5 | — | |
BUKMSYYNNHEANR
|
6.7 | IC50 | 2 | — | |
CSCUXLKCEJASIE
|
6.7 | IC50 | 2 | — | |
FVOCMDWBLIDMCB
|
6.7 | IC50 | 2 | — | |
MORVKBRPZDOTCQ
|
6.7 | IC50 | 2 | — | |
PXGLIUGVLBRUBV
|
6.7 | IC50 | 3 | — | |
SEMYKOKZLGFZNB
|
6.7 | IC50 | 2 | — | |
SKDYZXWYDRSLQY
|
6.7 | IC50 | 2 | — | |
TZBQXXNSSCAVKT
|
6.7 | IC50 | 2 | — | |
UIJBTFOXBSSWCE
|
6.7 | IC50 | 2 | — | |
WJCNNHJXSAZOGM
|
6.7 | IC50 | 2 | Yes | |
ZXCAATWSTKTNHY
|
6.7 | IC50 | 2 | — | |
AOFJRBMLTUGMMP
|
6.7 | Ki | 12 | — | |
BGUQECPEELVHLW
|
6.7 | Ki | 3 | — | |
BSFNGHCTZDCQBF
|
6.7 | Ki | 93 | — | |
HCNIBOQWDVOZKF
|
6.7 | Ki | 26 | — | |
HMXWMMRCKSDFCV
|
6.7 | IC50 | 10 | Yes | |
HQXRVTFLFJNGAV
|
6.7 | IC50 | 2 | — | |
JJGSOVIZOMZMCS
|
6.7 | Ki | 35 | — | |
JXMYIDZREHNPDO
|
6.7 | Ki | 19 | — | |
KUVJIFPAOJEBMN
|
6.7 | IC50 | 3 | — | |
LFVVQRUJKSZURN
|
6.7 | IC50 | 3 | — | |
NBZRNTFURGGIML
|
6.7 | IC50 | 2 | — | |
NJPWCTYVEJIQBM
|
6.7 | Ki | 72 | — | |
NRSGWEVTVGZDFC
|
6.7 | Ki | 50 | — | |
PCTRICLZSMFSET
|
6.7 | IC50 | 4 | Yes | |
PNKALLUVKOKYHZ
|
6.7 | Ki | 32 | — | |
QFOMGFNHXREHSV
|
6.7 | IC50 | 3 | — | |
QYGMZFLXMWJYRJ
|
6.7 | Ki | 14 | — | |
RAPYFGJGASETOS
|
6.7 | Ki | 11 | — | |
SHENEEFOURUIBP
|
6.7 | Ki | 29 | — | |
SJCISSZWYLCABC
|
6.7 | IC50 | 3 | — | |
UAQJVFADAYIBGC
|
6.7 | Ki | 23 | — | |
UHWVXMZHHQZRCC
|
6.7 | IC50 | 2 | Yes | |
UJBJWYNPUOLFIZ
|
6.7 | Ki | 49 | — | |
WDVLOKNHMBINOL
|
6.7 | IC50 | 3 | — | |
XLJHIFICPVNHJG
|
6.7 | IC50 | 2 | Yes | |
ZGZVRPRSFXRGCF
|
6.7 | Ki | 76 | — | |
ZWRIWNSRFLBBOD
|
6.7 | IC50 | 3 | — | |
ZXLFIHLBHMLHFJ
|
6.7 | Ki | 31 | — | |
VIJMQSQDODLIHT
|
6.7 | IC50 | 3 | — |