Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKSQRGQNPZBVPP
|
6.8 | IC50 | 4 | — | |
NYXQIXYXIOVJPB
|
6.8 | IC50 | 2 | — | |
OADRBDVURCEKRP
|
6.8 | Ki | 44 | — | |
SHPFDGWALWEPGS
|
6.8 | Kd | 35 | — | |
SKKGEOIZBPJZLM
|
6.8 | Ki | 3 | — | |
TWZVBMXTDSNZLS
|
6.8 | Ki | 7 | — | |
VAHCPZHCLNBIBJ
|
6.8 | IC50 | 4 | — | |
VQPBIJGXSXEOCU
|
6.8 | Ki | 24 | — | |
WFHQLAWBICSWPO
|
6.8 | IC50 | 4 | — | |
WVZWFOGYDXWKPT
|
6.8 | Ki | 5 | Yes | |
ZMNWFTYYYCSSTF
|
6.8 | Ki | 18 | — | |
DMHQDPVKKNQNCV
|
6.8 | IC50 | 3 | — | |
JCDAVUJUCMYZTJ
|
6.8 | IC50 | 2 | — | |
PYIBJGHLGTVZLN
|
6.8 | IC50 | 2 | — | |
XLFNLJYGUOLEJS
|
6.8 | IC50 | 26 | — | |
YTALSCBTOISJNF
|
6.8 | IC50 | 2 | — | |
ZIJIMHMKDXTURQ
|
6.8 | IC50 | 6 | Yes | |
QKYQHNYADWTLSP
|
6.8 | IC50 | 3 | — | |
RXKUYZFBEMBYSF
|
6.8 | IC50 | 2 | — | |
AEBGAQZHEWUQER
|
6.8 | IC50 | 2 | — | |
GJOLOIJGOFZXST
|
6.8 | IC50 | 3 | — | |
HXAUJHZZPCBFPN
|
6.8 | IC50 | 4 | — | |
JMFBKXJSFCPIKB
|
6.8 | IC50 | 2 | — | |
UGPDJIJFANODJH
|
6.8 | IC50 | 12 | — | |
WHLKRBBRZJQSQQ
|
6.8 | IC50 | 2 | — | |
GVBXGRYWKSAQLW
|
6.8 | IC50 | 2 | — | |
RYSYVUSXNRKLCL
|
6.8 | IC50 | 2 | — | |
XSPGWDVICYATDA
|
6.8 | IC50 | 2 | — | |
ALBFRPATCDNTBG
|
6.8 | IC50 | 2 | — | |
HSHDMLKUROTFFL
|
6.8 | IC50 | 2 | — | |
IAMWPQBDRXGGEF
|
6.8 | IC50 | 2 | — | |
KTPMQAQBFZCIRN
|
6.8 | IC50 | 3 | — | |
RDNMFMKLAZWNLN
|
6.8 | IC50 | 2 | — | |
UNGUWAMCUZJLAS
|
6.8 | IC50 | 3 | — | |
XEZNBKVBTAWBBR
|
6.8 | IC50 | 2 | — | |
FAEQSQDLHPQOMI
|
6.7 | IC50 | 2 | — | |
FPKSFXFWECAIBR
|
6.7 | IC50 | 6 | Yes | |
GRKTXONMLYKNPL
|
6.7 | IC50 | 2 | — | |
ICYNJWIBQVTAKQ
|
6.7 | IC50 | 2 | — | |
ISYIJSJVYFOFPY
|
6.7 | IC50 | 2 | — | |
KAHHZLXTLVPZAC
|
6.7 | IC50 | 3 | Yes | |
RZBCOYUBQNCKGM
|
6.7 | IC50 | 3 | — | |
XVNFBGOMJAUCKO
|
6.7 | IC50 | 3 | — | |
YFBSBJBNKSZCLY
|
6.7 | IC50 | 4 | — | |
AMWMGVKJAYQHID
|
6.7 | IC50 | 2 | — | |
IAYJLHOAEWIYAY
|
6.7 | IC50 | 4 | Yes | |
IBWNGAFCNXNEDG
|
6.7 | Ki | 4 | Yes | |
QLPKEICBTKFRKM
|
6.7 | Ki | 4 | Yes | |
XLKQULZCNWBLGW
|
6.7 | IC50 | 3 | Yes | |
YHBWHSCISDHNCC
|
6.7 | IC50 | 4 | — |