Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XCNVQVQBCBXNAC
|
6.9 | IC50 | 2 | — | |
CCIYHYFLYIQCJR
|
6.9 | IC50 | 3 | Yes | |
DVLIQRGISIJWEA
|
6.9 | IC50 | 2 | — | |
DWBNOASTWMOBSP
|
6.9 | IC50 | 2 | — | |
JDNWHCLQTRJTAJ
|
6.9 | IC50 | 6 | Yes | |
OBWNXGOQPLDDPS
|
6.9 | IC50 | 6 | Yes | |
PQNWGLHBIINSDV
|
6.9 | IC50 | 2 | — | |
QDTOATMXXSCADG
|
6.9 | IC50 | 2 | — | |
SRYOUBCWZIVZBY
|
6.9 | IC50 | 2 | — | |
WZSQZESQWZLUNN
|
6.9 | IC50 | 2 | — | |
AJZIGZOVWAFSBH
|
6.9 | IC50 | 2 | — | |
OJBKYYOYGSVDKS
|
6.9 | IC50 | 2 | — | |
CJFROAYTGUAJIP
|
6.8 | IC50 | 2 | — | |
NYKVYBKVQOVZIQ
|
6.8 | Ki | 2 | — | |
OEDBLXPEGILSSQ
|
6.8 | IC50 | 2 | — | |
PLAVWQHGBMTMFR
|
6.8 | IC50 | 2 | — | |
YAEXRFPBDXLXMG
|
6.8 | IC50 | 3 | — | |
ZJJLQRJTKOYJNO
|
6.8 | IC50 | 2 | — | |
DLZFRDYBPCZDDU
|
6.8 | IC50 | 2 | — | |
DONQOOXVVSQFSF
|
6.8 | IC50 | 2 | — | |
FNBGPMNXEGPANM
|
6.8 | Ki | 2 | Yes | |
IESKIIZEQNQSBR
|
6.8 | IC50 | 2 | — | |
IHGGWEBRARGZIY
|
6.8 | IC50 | 2 | — | |
INFCIXXPAUHEET
|
6.8 | Kd | 2 | — | |
KWNQIKSDUIQHRX
|
6.8 | IC50 | 2 | — | |
MZYVNBWBWMPZHH
|
6.8 | IC50 | 2 | — | |
NZEUGQYGRHEHEG
|
6.8 | IC50 | 3 | — | |
VDBPPXVERWJWQR
|
6.8 | IC50 | 2 | — | |
VQRJYECHVOWPDV
|
6.8 | IC50 | 6 | Yes | |
OZGUGQSGXNMCNT
|
6.8 | IC50 | 3 | — | |
DRKOUHSEDVEHEG
|
6.8 | IC50 | 3 | Yes | |
GHKMIOAEPALCFS
|
6.8 | IC50 | 6 | — | |
NHMACPMXYHTADL
|
6.8 | Ki | 3 | Yes | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
RQMVMSIAPOLUTD
|
6.8 | IC50 | 2 | — | |
VTCVDQBVMWVWLM
|
6.8 | IC50 | 2 | — | |
VFMJIULPVNSAOD
|
6.8 | IC50 | 3 | Yes | |
VFMJIULPVNSAOD
|
6.8 | IC50 | 2 | — | |
WTQDVZNJLFUQDW
|
6.8 | IC50 | 2 | — | |
ZWGGSMUWSPJJIU
|
6.8 | IC50 | 2 | — | |
APUCFXHENVUXCY
|
6.8 | Ki | 15 | — | |
AXIVWWPYPSYJLD
|
6.8 | Ki | 7 | Yes | |
CGFXXKQAUTXPSO
|
6.8 | IC50 | 2 | — | |
GAMJJHMLLXIWRZ
|
6.8 | IC50 | 4 | Yes | |
GZAJLQWXDGQIMQ
|
6.8 | IC50 | 2 | — | |
IZAVTOABECKIDH
|
6.8 | Ki | 20 | — | |
KNACLJBHKVSTDL
|
6.8 | Ki | 40 | — | |
KSJOLPSCOYLXKR
|
6.8 | IC50 | 2 | — | |
LKUJDAHYLPICSE
|
6.8 | Ki | 24 | — | |
MHWHPWMWKYXCRJ
|
6.8 | Ki | 32 | — |