Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DMWCSOYJGHLVEB
|
6.9 | IC50 | 2 | — | |
HEUMDSXNTRSQHK
|
6.9 | IC50 | 3 | Yes | |
KLMNDRZFWQDVRL
|
6.9 | IC50 | 3 | Yes | |
LPIMYXVAEGCNPJ
|
6.9 | Ki | 3 | Yes | |
NIWBUWMZKOEJTN
|
6.9 | IC50 | 7 | — | |
PIQNNSKBFMKWGB
|
6.9 | IC50 | 4 | Yes | |
YFNWWNRZJGMDBR
|
6.9 | Kd | 35 | — | |
YGEQQFLMLXRDQK
|
6.9 | IC50 | 3 | — | |
ZFOPWBXSJXQVFA
|
6.9 | IC50 | 3 | Yes | |
ZOKVMFNJBPBZCE
|
6.9 | IC50 | 7 | — | |
ZXVWACUTSNFQBK
|
6.9 | IC50 | 2 | — | |
CODJRIKNYSCBSA
|
6.9 | IC50 | 3 | — | |
FQSHTSWWNWIELG
|
6.9 | IC50 | 3 | — | |
JXDMCBSKXVYKEG
|
6.9 | IC50 | 2 | — | |
QKKIWEILHCXECO
|
6.9 | IC50 | 24 | — | |
AYJBHLUSGLQYDG
|
6.9 | Ki | 16 | — | |
BOBGABAXWFYHQX
|
6.9 | Ki | 9 | — | |
BTHLNBWTKKAULX
|
6.9 | Ki | 16 | — | |
DKZYXHCYPUVGAF
|
6.9 | Kd | 112 | — | |
GHPFQRTVUDXWCC
|
6.9 | Ki | 35 | — | |
HCNZXJZRFQSKII
|
6.9 | IC50 | 2 | — | |
IRLYGKITXNMDSM
|
6.9 | Ki | 2 | — | |
JAMDNXUAYUHJLJ
|
6.9 | Ki | 40 | — | |
MADCXGNPDBWPLM
|
6.9 | Ki | 25 | — | |
NXNQLECPAXXYTR
|
6.9 | Ki | 29 | — | |
PROLIXHVRCJEFH
|
6.9 | Ki | 46 | — | |
TVUWQDLBEOZVOU
|
6.9 | Ki | 41 | — | |
TYGGXVLXMOVTBS
|
6.9 | IC50 | 2 | — | |
UOOZSMNSBYVUGZ
|
6.9 | Ki | 32 | — | |
UPPGGRZNGRFDAU
|
6.9 | Ki | 21 | — | |
WFTZMAAMCVPJJT
|
6.9 | Ki | 26 | — | |
ZLVOTRRGLSDLPF
|
6.9 | Ki | 36 | — | |
AIQJXTOEZSDXHV
|
6.9 | IC50 | 3 | Yes | |
ARLBCCDWOPSKDJ
|
6.9 | IC50 | 3 | — | |
COYIMHAMNHOPTJ
|
6.9 | IC50 | 3 | — | |
ISVKXCPIKLZVQW
|
6.9 | IC50 | 3 | Yes | |
JNCRJZQZLMYLLM
|
6.9 | IC50 | 3 | Yes | |
JYTYZRSXADUJAY
|
6.9 | IC50 | 2 | — | |
KOLMPPLMZOKCEL
|
6.9 | IC50 | 3 | — | |
LEJNMWZPQMLOST
|
6.9 | IC50 | 3 | Yes | |
LYFBDMFXIXDJSD
|
6.9 | IC50 | 5 | Yes | |
MCVWAVHQVAZAKZ
|
6.9 | IC50 | 3 | — | |
OETFNYXAELUUOC
|
6.9 | IC50 | 5 | — | |
OGNYUTNQZVRGMN
|
6.9 | IC50 | 16 | Yes | |
QRFIOQPCVMNZPT
|
6.9 | IC50 | 3 | Yes | |
RETUSTLIJKZUGV
|
6.9 | IC50 | 5 | Yes | |
RGGYJEYZTPRESN
|
6.9 | IC50 | 6 | Yes | |
WOSUZOOSGPAWAC
|
6.9 | IC50 | 3 | — | |
GLSXPVFPHBFULR
|
6.9 | IC50 | 2 | — | |
IRGAIDAWHGYOKD
|
6.9 | IC50 | 5 | — |