Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QSIAXFKUFXOHHK
|
7.0 | IC50 | 5 | Yes | |
QYFQPPSZJOXIML
|
7.0 | Ki | 3 | — | |
RYEJQIGGOAKPKK
|
7.0 | IC50 | 3 | — | |
SCANZEHBHPIJEQ
|
7.0 | IC50 | 2 | Yes | |
SRROIPFGGDHJCJ
|
7.0 | Ki | 7 | — | |
UAUJVWLUSNTVTA
|
7.0 | IC50 | 6 | — | |
UDFDIIVNIYWXDM
|
7.0 | Ki | 74 | — | |
UHYYTYYLATYSHI
|
7.0 | IC50 | 2 | — | |
VHWZYWCQBINXOX
|
7.0 | Ki | 3 | — | |
VUMVSNOKSXZEBS
|
7.0 | IC50 | 2 | — | |
XFIFRGSEYNEXIW
|
7.0 | IC50 | 2 | — | |
XHHRGYCOEVNAKV
|
7.0 | Ki | 6 | Yes | |
XYZNKCSDQRKAFR
|
7.0 | Ki | 53 | — | |
YDPCOTOJRODRFO
|
7.0 | IC50 | 3 | — | |
QMPJPNBXRYVKQU
|
7.0 | IC50 | 2 | — | |
WVLFHLOAIDRNCV
|
7.0 | IC50 | 2 | — | |
YGXXXNQYDYUAKU
|
7.0 | IC50 | 2 | — | |
AHFWDQSNXFITEU
|
7.0 | Ki | 4 | Yes | |
LVYXERPKYAQGKM
|
7.0 | IC50 | 4 | — | |
YECBARDDCVULIS
|
7.0 | IC50 | 2 | — | |
GZCREURYZWXRHS
|
7.0 | IC50 | 6 | — | |
HTLXWQIMRWWAEB
|
7.0 | IC50 | 3 | — | |
YQQWGLNBSUZDRG
|
7.0 | IC50 | 2 | — | |
BNYXRPMABDQJJR
|
7.0 | Kd | 5 | — | |
BOAKEOMCZWRBDF
|
7.0 | IC50 | 3 | — | |
BOWWSMXUIIXBOU
|
7.0 | IC50 | 3 | Yes | |
CXQHYVUVSFXTMY
|
7.0 | Kd | 154 | — | |
FIAJCYVGOYDLFU
|
7.0 | IC50 | 3 | — | |
HBGNZQRVHBIHPS
|
7.0 | IC50 | 6 | Yes | |
HFLGPAUKVFOIOT
|
7.0 | IC50 | 4 | Yes | |
HFTUUUTZQAVFBK
|
7.0 | IC50 | 3 | Yes | |
IJXKSFMGCXZEEN
|
7.0 | IC50 | 3 | Yes | |
KRUCYZFEUFVOHN
|
7.0 | IC50 | 3 | Yes | |
MMCKCGTUACUYFW
|
7.0 | IC50 | 3 | — | |
NHHQJBCNYHBUSI
|
7.0 | IC50 | 220 | — | |
ODIUNKSOMOLOOF
|
7.0 | IC50 | 3 | — | |
YIGOVOVHNMDCGU
|
7.0 | IC50 | 3 | — | |
FYDMEKZWCPHGNB
|
7.0 | IC50 | 2 | — | |
HLESTJFKZRMHRR
|
7.0 | IC50 | 2 | — | |
IKENQUDOTQBCJH
|
6.9 | IC50 | 18 | — | |
KMWZKNHCFZNBFL
|
6.9 | Ki | 3 | Yes | |
WIYXOIDCQNFVET
|
6.9 | IC50 | 3 | — | |
YCQBFDHXDTYLME
|
6.9 | IC50 | 2 | — | |
YIEKEILDJWQXRB
|
6.9 | IC50 | 4 | — | |
JISRCHCXKMPPJP
|
6.9 | IC50 | 2 | — | |
SCIOAYVRXBCGMK
|
6.9 | IC50 | 2 | — | |
SCMNVDCXNVNNAF
|
6.9 | IC50 | 2 | — | |
SRKLAYWRZKLNHC
|
6.9 | IC50 | 3 | — | |
ZATGFXTWDKIEKC
|
6.9 | IC50 | 8 | Yes | |
AHUJBJSHCSTRQK
|
6.9 | IC50 | 2 | — |