Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RILOFFQNUDZMEB
|
7.1 | IC50 | 3 | — | |
RKEDDEYMKFGVCU
|
7.1 | Ki | 2 | — | |
TYNGHODBFDMDKR
|
7.1 | IC50 | 3 | — | |
ZUOHNZIRNKHHJE
|
7.1 | Ki | 3 | Yes | |
CGQAJNWPJQOPOT
|
7.1 | IC50 | 3 | — | |
COBLQYUYOHSZOW
|
7.1 | IC50 | 2 | Yes | |
ODXLGPSRHTWRAQ
|
7.1 | IC50 | 2 | — | |
RHDBNLYQAOUIAE
|
7.1 | IC50 | 2 | Yes | |
XBGNBDWNHXZVQA
|
7.1 | IC50 | 3 | — | |
XEUIIWAFFDHEEJ
|
7.1 | IC50 | 2 | — | |
HZHFVDKWMSMXTO
|
7.1 | IC50 | 2 | — | |
QRDCBCOPUDYBCB
|
7.1 | IC50 | 4 | — | |
SPVMVDXYFVXTKJ
|
7.1 | IC50 | 2 | — | |
ULZISYPWXIGTKR
|
7.1 | IC50 | 2 | Yes | |
YYLKKYCXAOBSRM
|
7.1 | Kd | 191 | — | |
DCKMTGBFLNPJPS
|
7.0 | IC50 | 4 | Yes | |
GYJAQAMQCBBAPY
|
7.0 | IC50 | 2 | — | |
ORGQNRJTEJDZTI
|
7.0 | IC50 | 2 | — | |
SWOMTHLQJFJUKX
|
7.0 | IC50 | 2 | — | |
WZTHBTBWYVSGPF
|
7.0 | IC50 | 4 | Yes | |
ZLHFILGSQDJULK
|
7.0 | IC50 | 37 | Yes | |
JVAFTPDILUBIGR
|
7.0 | IC50 | 9 | Yes | |
NOHJLJNUPONZRF
|
7.0 | IC50 | 3 | — | |
NYFLTGXJAHDIGK
|
7.0 | IC50 | 2 | — | |
ORCUWBLKOFIGIQ
|
7.0 | IC50 | 2 | — | |
VGWGJPGDBLUSNW
|
7.0 | IC50 | 3 | — | |
VTTYFSMWRGIKFX
|
7.0 | IC50 | 2 | — | |
ZXMSLCHJMUQKLG
|
7.0 | IC50 | 2 | — | |
HYDSSXBBNYALNP
|
7.0 | IC50 | 5 | — | |
IUTUNANTVVQXCT
|
7.0 | IC50 | 2 | — | |
IYBGHBZUXSMOKI
|
7.0 | IC50 | 3 | — | |
JUWVGQDRIAVTIK
|
7.0 | IC50 | 3 | — | |
QZCMKSLZWAYEFU
|
7.0 | IC50 | 2 | Yes | |
GXKIHPXGVQZMIN
|
7.0 | IC50 | 3 | — | |
ROJRDYDJKQGLRH
|
7.0 | IC50 | 3 | — | |
DPEWXXLKQMQEFN
|
7.0 | IC50 | 2 | — | |
JZUMLGZEZIDAPY
|
7.0 | IC50 | 2 | — | |
UVGSPPQDSXBTJW
|
7.0 | IC50 | 2 | Yes | |
AKWLDQDWZNJYKL
|
7.0 | IC50 | 14 | — | |
CAMXHQIJVZTBFW
|
7.0 | IC50 | 2 | — | |
CAQRLZFEWBTCCO
|
7.0 | IC50 | 3 | Yes | |
FZYXCINEILQJBV
|
7.0 | Ki | 2 | — | |
GBOGGRLNGKRGBK
|
7.0 | IC50 | 2 | — | |
GNMMAGUTRIXXSA
|
7.0 | IC50 | 2 | — | |
KCKXYZOBGBJZEG
|
7.0 | Ki | 36 | — | |
KXMZDGSRSGHMMK
|
7.0 | IC50 | 14 | — | |
KXPWWMPXNUOYOH
|
7.0 | Ki | 24 | — | |
MGGBYMDAPCCKCT
|
7.0 | Kd | 23 | — | |
MKAHLUQCHFLGCS
|
7.0 | IC50 | 2 | — | |
NJBJRWXJKAMYFV
|
7.0 | IC50 | 2 | — |