Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JBOORGPMLIAKTP
|
7.2 | IC50 | 3 | — | |
GVMDVMPNOAVKJR
|
7.1 | Ki | 26 | Yes | |
JRJLSKJAGSYHAP
|
7.1 | IC50 | 3 | — | |
KUVCMYWUDJSYSW
|
7.1 | IC50 | 2 | — | |
JUSQZYXEYZPLCG
|
7.1 | IC50 | 2 | Yes | |
AKIIIZOJWRPEPQ
|
7.1 | IC50 | 5 | Yes | |
BTWBYAOFMFQYSZ
|
7.1 | IC50 | 3 | — | |
DFAKFCGQJSYCEP
|
7.1 | IC50 | 2 | Yes | |
HRBFUNRZFJWHLJ
|
7.1 | IC50 | 2 | — | |
KLIDFKYRDXZCOP
|
7.1 | IC50 | 4 | — | |
KTEIFNKAUNYNJU
|
7.1 | Kd | 114 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
NIVIVGADJDEGJO
|
7.1 | IC50 | 2 | — | |
MRITYVDXXFOOAU
|
7.1 | Kd | 6 | — | |
SRNHAKVSFVSSPN
|
7.1 | IC50 | 8 | Yes | |
VNBRGSXVFBYQNN
|
7.1 | IC50 | 22 | Yes | |
DMKUCUYQRJKWJF
|
7.1 | Ki | 3 | — | |
DVROHIHHTSFVPB
|
7.1 | IC50 | 2 | — | |
HCKGGEPGRAIKER
|
7.1 | IC50 | 2 | — | |
HECCNHYZTOZRLV
|
7.1 | IC50 | 2 | Yes | |
HLXBUKYOKGQEDD
|
7.1 | IC50 | 2 | — | |
HTVKDECMTMXAPH
|
7.1 | IC50 | 5 | — | |
JSDGKSMNPHJDFK
|
7.1 | Ki | 35 | — | |
JXKDTYDBDDKIPY
|
7.1 | IC50 | 5 | Yes | |
KWSZYBNXNYRQCC
|
7.1 | Ki | 21 | — | |
MIJMZVTYIXYSDK
|
7.1 | Ki | 4 | — | |
MKAHLUQCHFLGCS
|
7.1 | IC50 | 2 | — | |
NJBJRWXJKAMYFV
|
7.1 | IC50 | 2 | — | |
NUALOIMAZAHWKR
|
7.1 | IC50 | 2 | — | |
OPLHMHMCXQXEQG
|
7.1 | Ki | 10 | — | |
QVMGDDAULZLNOQ
|
7.1 | Ki | 3 | — | |
RESQIOFIUHXDCZ
|
7.1 | IC50 | 2 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
RQIHWUXZUCCRLQ
|
7.1 | IC50 | 2 | — | |
RTDSHUGNRVXRHN
|
7.1 | Ki | 51 | — | |
WKMYUHUMKWPSCQ
|
7.1 | Ki | 3 | — | |
XCHWBXBDZRJVDP
|
7.1 | Ki | 51 | — | |
XDTMWNUVKUHOQV
|
7.1 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.1 | IC50 | 64 | Yes | |
XSDJOIOVIMPMHD
|
7.1 | Ki | 44 | — | |
YDOPLCNFRXOHCC
|
7.1 | Ki | 28 | — | |
CEAQTTJXUPADGI
|
7.1 | IC50 | 3 | Yes | |
CSIWGLJKPPOVQR
|
7.1 | Ki | 3 | Yes | |
CZBLMYRJPRLVRE
|
7.1 | IC50 | 3 | — | |
LCNZVWVKIFPDPM
|
7.1 | IC50 | 3 | Yes | |
MKPGJKRDMWXJIV
|
7.1 | IC50 | 2 | — | |
QZCMKSLZWAYEFU
|
7.1 | IC50 | 2 | Yes | |
FOANSKGMQAGOIR
|
7.1 | IC50 | 2 | — | |
JGBVPRGLWQWHIG
|
7.1 | IC50 | 2 | — | |
RDIZFHYTFVBBCX
|
7.1 | IC50 | 2 | Yes |