Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWYNGONSCKJMOW
|
7.2 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.2 | Kd | 147 | Yes | |
DIGPGAQNZZWPSG
|
7.2 | IC50 | 3 | Yes | |
IZZAJZCFAZXNDC
|
7.2 | IC50 | 6 | Yes | |
NACVPONJWZPHAP
|
7.2 | IC50 | 5 | Yes | |
OAIDOYYRSBXKJG
|
7.2 | IC50 | 3 | Yes | |
OAJNZHZQLRZZSC
|
7.2 | IC50 | 3 | Yes | |
RDFBXLTVSCZKAQ
|
7.2 | IC50 | 2 | — | |
CVMUHXWSBHMVGZ
|
7.2 | IC50 | 6 | Yes | |
FDZBZSBLRVVIGJ
|
7.2 | IC50 | 2 | — | |
FUSGHFKTWQRWPV
|
7.2 | Ki | 4 | — | |
GALVWTFFXPRMQM
|
7.2 | Ki | 20 | — | |
GLMWKEAUVZDGKE
|
7.2 | Ki | 23 | — | |
GTMDZIKJMWLLBV
|
7.2 | Ki | 3 | — | |
HEUSUIRCBWROMH
|
7.2 | Ki | 64 | — | |
JVAFTPDILUBIGR
|
7.2 | IC50 | 7 | — | |
KNGBPOUPNSUJPG
|
7.2 | IC50 | 2 | — | |
LCGSWTFWYNYUKS
|
7.2 | Ki | 26 | — | |
LQVXSNNAFNGRAH
|
7.2 | IC50 | 33 | Yes | |
MZDKLVOWGIOKTN
|
7.2 | Ki | 80 | — | |
NHUSXSLUEKKDFF
|
7.2 | IC50 | 2 | Yes | |
SPMHGQZFMNZCBV
|
7.2 | Ki | 30 | Yes | |
WZFYELPFTNDMJW
|
7.2 | IC50 | 2 | — | |
ZHNDVKCPJRLARD
|
7.2 | Ki | 3 | — | |
HEUIHAJXEGXNNB
|
7.2 | IC50 | 2 | Yes | |
LDGOZDNOQAZRQV
|
7.2 | IC50 | 2 | — | |
LHDNLQKQBSMXMU
|
7.2 | IC50 | 2 | — | |
NZJCXRPMZJGVCC
|
7.2 | Kd | 8 | — | |
UNYZXVQYBXGDJS
|
7.2 | IC50 | 2 | Yes | |
WMBJPWPAQLGSFL
|
7.2 | IC50 | 6 | Yes | |
XTOHRNRFRAUJKC
|
7.2 | IC50 | 3 | — | |
CBLIPXTZSVBWET
|
7.2 | IC50 | 3 | Yes | |
FFNIWOOLZGAOAB
|
7.2 | IC50 | 8 | Yes | |
OJFKUJDRGJSAQB
|
7.2 | IC50 | 17 | — | |
PQYSCCATMNNHGY
|
7.2 | IC50 | 2 | — | |
QZOGIXIGMUOFQB
|
7.2 | IC50 | 2 | — | |
WEGHHPFXCHFJFR
|
7.2 | Ki | 3 | — | |
ZEVUIDOBQPKBIO
|
7.2 | IC50 | 2 | — | |
IICOWTOEYHWWOH
|
7.2 | IC50 | 3 | — | |
MYMJRZXUXNYPIX
|
7.2 | IC50 | 2 | — | |
XIFWZYQJCXOJDM
|
7.2 | IC50 | 3 | — | |
BMYPVSWCQCKWHI
|
7.2 | IC50 | 3 | — | |
FYWNMALNWQLLBJ
|
7.2 | IC50 | 2 | — | |
HTHISIOYCCJIBY
|
7.2 | IC50 | 2 | — | |
KZBSEJKXWKPCLO
|
7.2 | Kd | 2 | — | |
WTSZLPJRFYTKQX
|
7.2 | IC50 | 2 | — | |
XGDJUMSXIASBOC
|
7.2 | IC50 | 2 | — | |
ASHFSDTVSQCVQC
|
7.2 | IC50 | 2 | — | |
CQOOBCLBMYGVDE
|
7.2 | IC50 | 3 | — | |
IRCOUATYCJGYHC
|
7.2 | IC50 | 2 | — |