Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WYOMXSAYYXBPMN
|
7.3 | Ki | 24 | — | |
XKZINYYXWJEYEL
|
7.3 | IC50 | 37 | — | |
XYXLUJQBBIBJFV
|
7.3 | Ki | 36 | — | |
YGJKHDBRTOPTNK
|
7.3 | Ki | 8 | — | |
ZWVZORIKUNOTCS
|
7.3 | Ki | 69 | — | |
CIXLLNNDLZVHIJ
|
7.3 | IC50 | 2 | — | |
FLGUGRAWIWHCJF
|
7.3 | IC50 | 4 | — | |
JJOKOLOYQZIVJV
|
7.3 | IC50 | 2 | — | |
JQTJXXKLVJKNLC
|
7.3 | IC50 | 2 | Yes | |
QHNJBHCDCYTMNB
|
7.3 | IC50 | 3 | Yes | |
UZFYLZWGFGEELR
|
7.3 | IC50 | 3 | — | |
VWQOMDPIYKNCFJ
|
7.3 | IC50 | 3 | Yes | |
XLXSRNTZHMLTMP
|
7.3 | Ki | 3 | Yes | |
GBXVVXZXFOFHSU
|
7.3 | Ki | 3 | Yes | |
GJFJLQXYFZSVOD
|
7.3 | IC50 | 2 | — | |
NEYBSPWSNSHKHW
|
7.3 | IC50 | 3 | — | |
OSVOVHIYXDNBJQ
|
7.3 | IC50 | 3 | — | |
PIBTTWIAIOIVKG
|
7.3 | IC50 | 2 | — | |
XUTDOIHRJBCEMW
|
7.3 | IC50 | 2 | — | |
DVDNHJJINLEZSO
|
7.3 | IC50 | 3 | — | |
MFWHDFGMXHATNR
|
7.3 | IC50 | 3 | — | |
NVJBRKUSNQZNKX
|
7.3 | IC50 | 3 | Yes | |
SOTHNRIRXPUQEZ
|
7.3 | IC50 | 5 | Yes | |
AKSIZPIFQAYJGF
|
7.3 | IC50 | 4 | Yes | |
NYPQIYNAJRTAPS
|
7.3 | IC50 | 3 | — | |
OKKAENUKIYEBBD
|
7.3 | IC50 | 4 | Yes | |
FJZFOTKMZCYJDF
|
7.2 | IC50 | 4 | — | |
HNXLEVKZEPXIAQ
|
7.2 | IC50 | 2 | — | |
OXCBIRNMZPQWLB
|
7.2 | IC50 | 2 | Yes | |
RAOIIZFWMFAGEK
|
7.2 | IC50 | 2 | — | |
VIHXUAKPZPXVSW
|
7.2 | IC50 | 6 | Yes | |
ATUGFOWGVANOHQ
|
7.2 | Ki | 4 | Yes | |
BTQCPHBDUJMLMF
|
7.2 | IC50 | 2 | Yes | |
DYTKVFHLKPDNRW
|
7.2 | Ki | 23 | Yes | |
GAAHSFKFIMENOG
|
7.2 | IC50 | 3 | Yes | |
HFSFBCFFSSYGFK
|
7.2 | IC50 | 3 | Yes | |
IRGIWNWHHPMOLO
|
7.2 | IC50 | 3 | — | |
OYPSWGQEIRWPRG
|
7.2 | IC50 | 2 | — | |
RPSFIQJOUUTWRS
|
7.2 | IC50 | 3 | Yes | |
WZOYNDVCXZRUFV
|
7.2 | IC50 | 3 | — | |
AGHMFEHJWZVACU
|
7.2 | Ki | 3 | Yes | |
HZUXHEBYLGLOGZ
|
7.2 | IC50 | 2 | — | |
NQHMMDRPRXVCLT
|
7.2 | IC50 | 8 | Yes | |
PZWGYFJPWNXLGT
|
7.2 | IC50 | 3 | — | |
XTWXMJDVQOEURD
|
7.2 | IC50 | 3 | Yes | |
AEINMBOZWWDMIV
|
7.2 | IC50 | 3 | — | |
DQRVOAFQMMLWCP
|
7.2 | IC50 | 3 | — | |
KJAGZTFLBMDQQT
|
7.2 | IC50 | 3 | Yes | |
OZWMSXPIQVMFDE
|
7.2 | IC50 | 8 | Yes | |
VCLDLBGMMXCQJL
|
7.2 | IC50 | 3 | — |