Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SKDSRJRRAQLUPP
|
7.3 | IC50 | 8 | Yes | |
UEIDWGGSGUODLX
|
7.3 | IC50 | 2 | — | |
VCBGNDQGKNIBBK
|
7.3 | IC50 | 6 | Yes | |
XXHKWYBEHKUWRK
|
7.3 | IC50 | 2 | — | |
YOZAGBCKIMCHID
|
7.3 | IC50 | 3 | Yes | |
BEVPJXUTHBNTLS
|
7.3 | IC50 | 3 | Yes | |
FHSKCOBLBQSSQE
|
7.3 | IC50 | 3 | Yes | |
IRGAVEDIAARWCQ
|
7.3 | IC50 | 2 | — | |
OUEYXPDIZLXCBG
|
7.3 | IC50 | 3 | Yes | |
SKNITDPTVHFEGL
|
7.3 | IC50 | 2 | Yes | |
NHFDRBXTEDBWCZ
|
7.3 | IC50 | 12 | Yes | |
SBSYQSASKXLENU
|
7.3 | IC50 | 5 | Yes | |
SIRZTYWYVGTPEV
|
7.3 | IC50 | 4 | — | |
UDKDYWHGVWVLDY
|
7.3 | IC50 | 3 | Yes | |
AKJBLKUZXRMECW
|
7.3 | Kd | 6 | — | |
BNCDEGOHMGKVSC
|
7.3 | IC50 | 2 | — | |
GFWYLCYLWSMJSC
|
7.3 | IC50 | 3 | — | |
KGHHVSJZWGWWDG
|
7.3 | IC50 | 4 | Yes | |
KVLWNTNKPNPJIZ
|
7.3 | IC50 | 2 | — | |
MOQBNQNUPNPLCH
|
7.3 | IC50 | 7 | Yes | |
OBVWAZKFFALEAF
|
7.3 | IC50 | 2 | — | |
RMJGEOPKVZZYTL
|
7.3 | IC50 | 2 | — | |
JOQPAKTWBKIHRT
|
7.3 | IC50 | 2 | — | |
PGYJINWZLJSDIT
|
7.3 | Ki | 2 | Yes | |
RBNRSVPXZPBXCD
|
7.3 | IC50 | 5 | — | |
SDEWZAPYGJGVJM
|
7.3 | IC50 | 2 | — | |
AKBNORYPCWJWFZ
|
7.3 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
7.3 | Ki | 55 | — | |
DKZGAIQFKXCKMJ
|
7.3 | IC50 | 2 | — | |
GAMJJHMLLXIWRZ
|
7.3 | IC50 | 3 | Yes | |
GJAFGIYDCWQVAO
|
7.3 | IC50 | 2 | — | |
HNGRKZKIRRQEDF
|
7.3 | IC50 | 3 | Yes | |
JUXJSIGKLXPRRY
|
7.3 | IC50 | 2 | Yes | |
JYNKKTHUZTYHCU
|
7.3 | Ki | 3 | — | |
KOHNRDPXFDZZJF
|
7.3 | Ki | 31 | — | |
KTEIFNKAUNYNJU
|
7.3 | Ki | 48 | — | |
LDGOZDNOQAZRQV
|
7.3 | IC50 | 2 | — | |
MPSOTLJRIZYQCG
|
7.3 | IC50 | 3 | — | |
NLUPJKQOKWBWFC
|
7.3 | Ki | 69 | — | |
QEJOFXISUMFQBD
|
7.3 | IC50 | 2 | — | |
QXRJBJVCBQSLTA
|
7.3 | Ki | 29 | — | |
RKKIDHHGKNGTQI
|
7.3 | Ki | 28 | — | |
UHPJJAZNFIBQPH
|
7.3 | IC50 | 2 | — | |
UXMNYFJHEBEDJS
|
7.3 | Ki | 19 | Yes | |
VFXRIBNDTAAKLH
|
7.3 | IC50 | 4 | — | |
VNDWQCSOSCCWIP
|
7.3 | Ki | 39 | Yes | |
VSVWQTDDGQSGHP
|
7.3 | Ki | 51 | — | |
WBQBMMMQJSJEJT
|
7.3 | Ki | 4 | — | |
WFOLLQWDLJNOGD
|
7.3 | IC50 | 2 | — | |
WHYSRBRRFPMZRT
|
7.3 | IC50 | 2 | Yes |