Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZJQWORQRPDYKRS
|
7.4 | IC50 | 7 | — | |
AWDORCFLUJZUQS
|
7.4 | Ki | 22 | — | |
CXBBWVXSZINRCS
|
7.4 | Ki | 41 | — | |
DCTBPIBEQFLAOQ
|
7.4 | Ki | 13 | — | |
FGBBAYDBFFBOCR
|
7.4 | IC50 | 2 | — | |
FXQWJULRETZHHW
|
7.4 | Ki | 14 | — | |
HWXNNRXRMBATRT
|
7.4 | IC50 | 2 | Yes | |
KLAOKWJLUQKWIF
|
7.4 | Ki | 5 | — | |
LWIAVJGVALWTGR
|
7.4 | IC50 | 2 | — | |
NPJROAJIXPVMTE
|
7.4 | Ki | 8 | — | |
NWMPVMMGSHXANZ
|
7.4 | Ki | 58 | — | |
RJLAEHDOQAMXKD
|
7.4 | IC50 | 2 | — | |
UQNNJYLAPYGZBD
|
7.4 | Ki | 28 | — | |
WRRLCKCZMMPCBS
|
7.4 | Ki | 3 | — | |
WUWDLXZGHZSWQZ
|
7.4 | Ki | 41 | — | |
WVFWTUJEHMVUBG
|
7.4 | Ki | 25 | — | |
YQEBSIBQRPFUBN
|
7.4 | IC50 | 3 | — | |
YQWYJLZXGVWBRR
|
7.4 | Ki | 2 | — | |
ZAARMHXLYCHRAK
|
7.4 | Ki | 20 | — | |
DFIKQTZUHIIMDU
|
7.4 | IC50 | 2 | — | |
GANVFRXETVPEAB
|
7.4 | IC50 | 2 | — | |
KBJCTAIADOTYHC
|
7.4 | IC50 | 8 | Yes | |
KGXBCWANASZZQG
|
7.4 | IC50 | 5 | — | |
KHDTZPRXPIQIDD
|
7.4 | IC50 | 3 | — | |
UFATYBRKMMRKGA
|
7.4 | Kd | 3 | — | |
WBOJNPOFWWQXBX
|
7.4 | IC50 | 4 | — | |
YQTIZDYSQKQTBQ
|
7.4 | IC50 | 2 | — | |
GEATXDJAPAHPTP
|
7.4 | IC50 | 10 | — | |
ROGHHIGHHTZCFT
|
7.4 | IC50 | 3 | Yes | |
RZLXGZULLYTTFO
|
7.4 | Ki | 3 | — | |
SROFNWNYOOAXPQ
|
7.4 | IC50 | 2 | — | |
AXMMFQYWZDPEFR
|
7.4 | IC50 | 2 | — | |
BLFRZPJRKJLHGU
|
7.4 | IC50 | 3 | — | |
HHFBDROWDBDFBR
|
7.4 | IC50 | 40 | Yes | |
KJMURTHIPWRIMC
|
7.4 | IC50 | 7 | — | |
SEJGTFPOEJWEGG
|
7.4 | Kd | 149 | — | |
UQXVKPUPDOHDDK
|
7.4 | IC50 | 3 | — | |
WOTWXKACTZFRQE
|
7.4 | IC50 | 4 | — | |
YLJVNDQEACKRKQ
|
7.4 | IC50 | 2 | — | |
ZJTCESMUJZZNAL
|
7.4 | IC50 | 3 | — | |
CSFNNUIZTRGKSQ
|
7.4 | IC50 | 3 | Yes | |
HJQMKDZFPSWOEL
|
7.4 | IC50 | 2 | — | |
NYHVIVWBHLTODF
|
7.4 | IC50 | 3 | Yes | |
PLJWNSJCDIUAGM
|
7.4 | IC50 | 2 | — | |
XNPFPPICVRIXSI
|
7.4 | IC50 | 2 | — | |
BOQOQFWDFXIKGR
|
7.3 | IC50 | 2 | — | |
DXXQAWREKCQJCS
|
7.3 | IC50 | 4 | — | |
GSMALWRBDKEIGI
|
7.3 | IC50 | 2 | — | |
ORWIYCURPDKSBI
|
7.3 | IC50 | 15 | Yes | |
ROPCWFYJUONUHM
|
7.3 | IC50 | 4 | — |