Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CFBXWHPXNROFFK
|
7.6 | IC50 | 4 | — | |
CZFUYZPXZGGWKC
|
7.6 | IC50 | 7 | — | |
DADASRPKWOGKCU
|
7.6 | IC50 | 9 | — | |
FJGYGQJTRHDGSL
|
7.6 | IC50 | 2 | — | |
HOCURELMRBRHRJ
|
7.6 | IC50 | 3 | — | |
KEZAFIAURWAGLZ
|
7.6 | IC50 | 3 | Yes | |
RAPHAQZUOBFENV
|
7.6 | IC50 | 6 | Yes | |
RWCPLVNQNAADEI
|
7.6 | IC50 | 2 | — | |
VMQIKSUBUKPMBA
|
7.6 | IC50 | 3 | Yes | |
KDKUVYLMPJIGKA
|
7.6 | IC50 | 91 | Yes | |
UEKBKVAQJQTBGW
|
7.6 | IC50 | 3 | — | |
DBXGGXLBTWZXBB
|
7.6 | Ki | 39 | — | |
FZTUPODAEPTYNG
|
7.6 | IC50 | 4 | Yes | |
GFHRPONHRZBFNC
|
7.6 | IC50 | 3 | — | |
IWKRMYPMEYTIEG
|
7.6 | Ki | 2 | — | |
JIJDOMRYZXJLMB
|
7.6 | IC50 | 2 | Yes | |
KVXXTWMZAGQKMI
|
7.6 | IC50 | 3 | — | |
LCVIRAZGMYMNNT
|
7.6 | IC50 | 20 | — | |
LILXUVCZUBSSFA
|
7.6 | IC50 | 6 | — | |
MENUIGPUGBMCMV
|
7.6 | IC50 | 2 | — | |
RHGZQGXELRMGES
|
7.6 | IC50 | 8 | Yes | |
SUIPNNKRHBDYHW
|
7.6 | IC50 | 2 | Yes | |
XACWBNSEGIFUIV
|
7.6 | IC50 | 3 | — | |
YUJACPUEEGUFHA
|
7.6 | IC50 | 3 | Yes | |
BSFSQSWHBCBLLD
|
7.6 | IC50 | 2 | — | |
MENIKIFJGYYVNI
|
7.6 | IC50 | 5 | Yes | |
MQWHYEKERKXFQY
|
7.6 | IC50 | 2 | — | |
NKQFVOKSVRQZKX
|
7.6 | IC50 | 2 | — | |
QBOWGZQRUNUQGL
|
7.6 | IC50 | 3 | — | |
SYOBTEQVKWAJIS
|
7.6 | IC50 | 2 | — | |
HLXBUKYOKGQEDD
|
7.6 | IC50 | 2 | — | |
HQTDBFXCCUUCFU
|
7.6 | IC50 | 2 | — | |
LLGYBOCRDSLEKE
|
7.6 | IC50 | 3 | Yes | |
MGHRIOSQJVOCSQ
|
7.6 | IC50 | 2 | — | |
NUPQKBHSBNJYIP
|
7.6 | IC50 | 2 | — | |
PWZXORMRRWDONZ
|
7.6 | IC50 | 3 | Yes | |
SMAYBYUGIIIPKY
|
7.6 | IC50 | 3 | Yes | |
VKVBESYYODLWDZ
|
7.6 | IC50 | 2 | — | |
XFHCSNRQFQRLHZ
|
7.6 | Ki | 12 | Yes | |
FURXQBPRWUDWOM
|
7.6 | IC50 | 2 | — | |
GFUZUEVAWXYASP
|
7.6 | IC50 | 3 | — | |
KFYFFELQRLSBEN
|
7.6 | IC50 | 2 | — | |
KHDLZWDZNAKTKK
|
7.6 | Ki | 4 | Yes | |
LTTWDGKJGMQNHP
|
7.6 | IC50 | 3 | — | |
RGXAJUCULIIOCG
|
7.6 | IC50 | 2 | — | |
VWNWNXCVJAUZBJ
|
7.6 | IC50 | 2 | — | |
ZUXFIRWLAQBCCS
|
7.6 | IC50 | 8 | Yes | |
SCMPDMAJYNSKMW
|
7.6 | IC50 | 3 | — | |
YRDHKIFCGOZTGD
|
7.6 | IC50 | 21 | — | |
APEKZEQPEXYFDS
|
7.5 | IC50 | 2 | — |