Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QLPWFQPHRAFDGC
|
7.7 | IC50 | 7 | — | |
SFXBHFZUSIUICI
|
7.7 | IC50 | 2 | — | |
UNXQVAHMAHJXJM
|
7.7 | IC50 | 3 | Yes | |
GXSLNZRYHCTIMQ
|
7.7 | IC50 | 2 | — | |
KRRYGFBABIBCHR
|
7.7 | IC50 | 3 | — | |
BNPHQQLNFFGRJU
|
7.7 | Ki | 2 | — | |
CKVWQORGCCEYHS
|
7.7 | Ki | 50 | — | |
CRVFIGQYZIENPM
|
7.7 | IC50 | 3 | Yes | |
DAIWPAQKPHJILU
|
7.7 | IC50 | 2 | — | |
GWMATETWMAQOFL
|
7.7 | Ki | 36 | — | |
HUIHLSDJNYBMSR
|
7.7 | Ki | 2 | — | |
LCQYMDMUCJFFKN
|
7.7 | IC50 | 5 | Yes | |
LRLDYTTWQIFWBD
|
7.7 | Ki | 25 | — | |
NECQZMQPXFYVOY
|
7.7 | Ki | 26 | — | |
NFMGZVPRGVERNN
|
7.7 | Ki | 44 | — | |
NHFDRBXTEDBWCZ
|
7.7 | Ki | 41 | — | |
QXNNCHKUKMPZRH
|
7.7 | IC50 | 2 | — | |
SDBOIBYRBWPIEL
|
7.7 | Ki | 31 | — | |
SJHNCEZKOYCERN
|
7.7 | Ki | 3 | — | |
VIDVOURISMXBLG
|
7.7 | IC50 | 3 | — | |
XLUIYTJCFLMYKF
|
7.7 | IC50 | 2 | — | |
ZVWRFVCNQOECJS
|
7.7 | Ki | 71 | — | |
DUAVMQAFJJEDTP
|
7.7 | IC50 | 3 | — | |
FJLUYTVEVSZLJP
|
7.7 | IC50 | 5 | — | |
ISOQIZINACKWNJ
|
7.7 | IC50 | 3 | — | |
LMSNQXFIZAHXQB
|
7.7 | IC50 | 3 | Yes | |
RQUYVPRGCIDFDN
|
7.7 | IC50 | 2 | — | |
UNRMMILBIIITEU
|
7.7 | IC50 | 3 | — | |
YQONVVWDOUUEGH
|
7.7 | IC50 | 2 | — | |
FYWIPSZJJOUPAR
|
7.7 | IC50 | 2 | — | |
IVVSNTYYOLGITN
|
7.7 | IC50 | 2 | — | |
IYCVFSSCAPZAJP
|
7.7 | IC50 | 5 | — | |
JPQQLLUZYXRSBP
|
7.7 | IC50 | 2 | Yes | |
KSFGFFQQMLCHJC
|
7.7 | IC50 | 3 | — | |
OPRMTHPWLRWOPL
|
7.7 | IC50 | 3 | — | |
PWTTWLQRFVOJIZ
|
7.7 | IC50 | 3 | Yes | |
RTWJZWFAMFOLDK
|
7.7 | IC50 | 2 | — | |
SCRSXZZGUOEUBI
|
7.7 | IC50 | 4 | Yes | |
XEXXLSSPQTWUID
|
7.7 | IC50 | 3 | — | |
XHXXOAPJDJYKTL
|
7.7 | IC50 | 2 | — | |
YXEIECLOAMHVCH
|
7.7 | IC50 | 3 | Yes | |
UMXZZNNMKDFYAG
|
7.7 | IC50 | 2 | — | |
BQYUDMQJOHMTEM
|
7.6 | IC50 | 3 | Yes | |
GOEHHWWOYYPDII
|
7.6 | IC50 | 6 | Yes | |
LEWVUPUKJSFGLR
|
7.6 | Ki | 3 | Yes | |
MJMJYGWCNKSGSI
|
7.6 | IC50 | 2 | — | |
OGDURDWHHQUSDO
|
7.6 | IC50 | 2 | — | |
PCBXYEMAQBQSOC
|
7.6 | IC50 | 3 | — | |
VCHQRSNNPYKZBM
|
7.6 | IC50 | 2 | — | |
WFRNKIOQSRRDQF
|
7.6 | IC50 | 3 | — |