Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NRDHAKDUAFEDCQ
|
7.8 | Ki | 3 | — | |
PMBSIXYFBNTLCB
|
7.8 | Ki | 2 | — | |
PXVPCLNOMYTQQA
|
7.8 | IC50 | 2 | — | |
QKPLUKMJEKRAJD
|
7.8 | Ki | 30 | Yes | |
RAEHGBLXUBDQLP
|
7.8 | IC50 | 4 | — | |
RBZINWUMPZNWCZ
|
7.8 | IC50 | 4 | Yes | |
RJZDECGDCKOHBV
|
7.8 | Ki | 70 | — | |
TWTUUCKVMANLPL
|
7.8 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes | |
UYJNQQDJUOUFQJ
|
7.8 | Ki | 68 | — | |
VBIFOMKCIFTINW
|
7.8 | IC50 | 4 | — | |
VCSQVKQFGYRGEH
|
7.8 | Ki | 13 | — | |
WHHJYUVJNITNFN
|
7.8 | IC50 | 4 | — | |
WRNRMZJJSTUZHL
|
7.8 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.8 | Ki | 56 | — | |
ZGDSBEUMPIMXBM
|
7.8 | Ki | 42 | — | |
STTWKDVRVDYNAH
|
7.8 | IC50 | 2 | — | |
SZJNVWAZUIGEQD
|
7.8 | IC50 | 2 | — | |
VYCUQEPITATEOI
|
7.8 | IC50 | 2 | — | |
AYHJBFRPPDPHQD
|
7.8 | IC50 | 2 | — | |
BTZIOWUABPKONC
|
7.8 | IC50 | 2 | — | |
GJSXBANTJATBDM
|
7.8 | IC50 | 2 | — | |
HEBQIUUCKUBQCJ
|
7.8 | IC50 | 2 | — | |
JBYKCUNHSBWUPW
|
7.8 | IC50 | 2 | — | |
PASPLONSFSXGKA
|
7.8 | IC50 | 2 | — | |
WANOQCJEBRGYPS
|
7.8 | IC50 | 3 | — | |
WEVRAOPLGYJTLY
|
7.8 | IC50 | 2 | — | |
XIZHRWKYFLKHBC
|
7.8 | IC50 | 4 | Yes | |
YEVNPJOHBLEPGC
|
7.8 | IC50 | 2 | — | |
VCRPHLZHPCWATH
|
7.8 | IC50 | 2 | — | |
CCMSKNPVKGYHGE
|
7.8 | IC50 | 3 | — | |
GCIKSSRWRFVXBI
|
7.8 | IC50 | 109 | Yes | |
AKBDTDXHGVXZLY
|
7.7 | IC50 | 4 | — | |
ARQPPPCSTGSCQR
|
7.7 | IC50 | 3 | Yes | |
ATZVMUKUKXZZAJ
|
7.7 | IC50 | 2 | — | |
BRVRJAZHVITNIF
|
7.7 | IC50 | 3 | Yes | |
CGEOTWGXFRJZLW
|
7.7 | IC50 | 3 | — | |
DEYRVWAAPWPOND
|
7.7 | IC50 | 3 | Yes | |
DLGIXSWHFYBLQG
|
7.7 | IC50 | 2 | — | |
GPWGVKOPIRJRKV
|
7.7 | Ki | 2 | — | |
MEWSLTZRULAUFE
|
7.7 | IC50 | 3 | Yes | |
OVSOFMFOYROLMC
|
7.7 | IC50 | 2 | — | |
QXTIKAMWRHHMBU
|
7.7 | IC50 | 3 | — | |
WUBFAXNVDMCVIO
|
7.7 | IC50 | 12 | Yes | |
MQWHYEKERKXFQY
|
7.7 | IC50 | 2 | — | |
VIVMIDXUVLTISY
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
IOUPQNBCPLQNGI
|
7.7 | IC50 | 3 | — | |
JWILUIVAYLRFIY
|
7.7 | IC50 | 14 | — | |
LOGJQOUIVKBFGH
|
7.7 | IC50 | 11 | Yes |