Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OMFRMSODXLGAQT
|
7.9 | IC50 | 3 | — | |
UWVYYAZEVUASFC
|
7.9 | IC50 | 3 | — | |
WAGMGFBPNPADDU
|
7.9 | IC50 | 2 | — | |
WGGOYMCUJRCWRJ
|
7.9 | IC50 | 3 | — | |
ZDDHVWIKFYVEKR
|
7.9 | IC50 | 3 | — | |
UVNLAMSMBMXIJB
|
7.9 | IC50 | 2 | — | |
GGLRONBKQRZFOT
|
7.9 | IC50 | 3 | — | |
ADTSCWGDALDZSK
|
7.8 | Ki | 2 | — | |
ANTUVUVMQSIJBS
|
7.8 | IC50 | 3 | Yes | |
AYVATFZLZLWIPA
|
7.8 | IC50 | 3 | — | |
HMLDXQBTXVPSOC
|
7.8 | IC50 | 3 | — | |
IBAUSYCHSXHDOA
|
7.8 | IC50 | 3 | — | |
IZDBEJJRNUSRIU
|
7.8 | IC50 | 3 | — | |
JJHXPDTVQKWKHA
|
7.8 | IC50 | 3 | Yes | |
FGKOFCQQLIEQOZ
|
7.8 | IC50 | 2 | — | |
PHENCDSAYZNXRO
|
7.8 | IC50 | 3 | — | |
XLSPYLMTRXPYKY
|
7.8 | IC50 | 13 | — | |
ADLPKFFMGIJZIM
|
7.8 | IC50 | 44 | — | |
AZRBHUUEXRGWFH
|
7.8 | Ki | 3 | — | |
CMEKRUHUVGTVLK
|
7.8 | IC50 | 6 | Yes | |
DKVKUPRCFKTRIY
|
7.8 | IC50 | 7 | — | |
DZICJKNDYKNBTO
|
7.8 | IC50 | 4 | Yes | |
IOGOXIFSMAQQPS
|
7.8 | IC50 | 2 | — | |
LBAGNMNWIAWTLK
|
7.8 | IC50 | 2 | — | |
MNGNUDIQTBWWNA
|
7.8 | IC50 | 3 | — | |
MVQSZXIVEQECJQ
|
7.8 | IC50 | 2 | — | |
NZSZVQMHSLFGDA
|
7.8 | IC50 | 2 | — | |
OQAVDYCSFNEKFW
|
7.8 | IC50 | 2 | — | |
PNQGVSADKMNRHP
|
7.8 | IC50 | 2 | — | |
QDKAHXFKNDNBHM
|
7.8 | IC50 | 2 | — | |
RKUJYVCXPDDJQR
|
7.8 | IC50 | 2 | — | |
RYROLHUONOCJPP
|
7.8 | IC50 | 2 | — | |
TWGQOAACISTFEJ
|
7.8 | IC50 | 2 | — | |
WKDACQVEJIVHMZ
|
7.8 | IC50 | 46 | — | |
YFLNJIAXYKROBA
|
7.8 | IC50 | 3 | — | |
ZLLVQOSTXBHAIP
|
7.8 | Ki | 3 | Yes | |
AIQDZMUPVYDVLB
|
7.8 | Ki | 48 | — | |
ATMONDFPCFVRCS
|
7.8 | IC50 | 3 | — | |
DZJJTOUVFUJWPC
|
7.8 | IC50 | 2 | — | |
FGSLHCMPNMYQJT
|
7.8 | Ki | 3 | — | |
HIXRSEFUZBICPP
|
7.8 | IC50 | 2 | — | |
HRZOUBQYVUXBNS
|
7.8 | Ki | 38 | — | |
IJHINRNPHQTGCM
|
7.8 | IC50 | 3 | — | |
ISVHLTLEHRZKJC
|
7.8 | Ki | 19 | — | |
JWFVSAJXAAUKIH
|
7.8 | IC50 | 2 | — | |
KVEIKKQFXLWWMV
|
7.8 | IC50 | 3 | — | |
LSEOXFVSQOHSDK
|
7.8 | Kd | 3 | — | |
MCCCQFAOMZMZKE
|
7.8 | IC50 | 52 | — | |
MWENAPMGLKQUOH
|
7.8 | IC50 | 2 | Yes | |
NFKMFNBKEOQNPZ
|
7.8 | Ki | 43 | — |