Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVBBUHNPXVGJKW
|
8.0 | IC50 | 2 | — | |
XSPXJYVALVHTAJ
|
8.0 | IC50 | 3 | — | |
BPCDCTRGBDOCQS
|
8.0 | IC50 | 2 | — | |
CITUHDBZOGJAEN
|
8.0 | IC50 | 3 | — | |
CXCXNZWXDOVZBA
|
8.0 | IC50 | 3 | — | |
DYBGLIINTRJUKT
|
8.0 | IC50 | 2 | — | |
KOOZPNYTOCFUNJ
|
8.0 | IC50 | 3 | — | |
KZBSEJKXWKPCLO
|
8.0 | IC50 | 3 | — | |
LHPRXXKFQZEGMG
|
8.0 | IC50 | 3 | Yes | |
NRGYZNJPCGRCLV
|
8.0 | IC50 | 52 | — | |
NRRLLJHNIQEBIO
|
8.0 | IC50 | 2 | — | |
OEYWYCKNHSHGIV
|
8.0 | IC50 | 2 | — | |
QCETXMLIFLYKQH
|
8.0 | IC50 | 3 | — | |
RITAVMQDGBJQJZ
|
8.0 | Kd | 43 | — | |
RYYNGWLOYLRZLK
|
8.0 | IC50 | 45 | — | |
VBWCCTREXYTDOA
|
8.0 | IC50 | 2 | — | |
XAQZJRAEQPCWMI
|
8.0 | Ki | 3 | Yes | |
CDBRRCRVKIRWPN
|
8.0 | IC50 | 2 | — | |
VKBFHTIUXUCYRQ
|
8.0 | IC50 | 8 | — | |
OJYFHTZIIPZQCE
|
7.9 | IC50 | 2 | — | |
YYFZPPMJHCVHFH
|
7.9 | IC50 | 2 | — | |
DUKZDMUZDDNVFF
|
7.9 | IC50 | 3 | — | |
FZVCMCRNWSWUCG
|
7.9 | IC50 | 3 | — | |
IZQYRTPRXYJMAX
|
7.9 | IC50 | 2 | — | |
NLGYPTWGAPKFAZ
|
7.9 | IC50 | 3 | — | |
NUIGAOCWJPYVEO
|
7.9 | IC50 | 2 | — | |
OTYSGQZTYQYLDD
|
7.9 | IC50 | 2 | — | |
RAVOJQLJGOGZMT
|
7.9 | IC50 | 2 | — | |
VNLDWMOEKZFKDP
|
7.9 | IC50 | 3 | — | |
XEXXLSSPQTWUID
|
7.9 | IC50 | 3 | — | |
YUAALFPUEOYPNX
|
7.9 | IC50 | 3 | — | |
YXMQIWJYPNBZJS
|
7.9 | IC50 | 4 | — | |
YXMQIWJYPNBZJS
|
7.9 | IC50 | 2 | — | |
ZGMGZBILRTWEQE
|
7.9 | IC50 | 2 | — | |
JFWCDNMTPZUMAD
|
7.9 | Ki | 2 | — | |
KKYPRNBBPBRJQX
|
7.9 | Ki | 40 | — | |
RWEHAHIEUDLKGT
|
7.9 | Ki | 33 | — | |
UQJQNZHGEVLHST
|
7.9 | Ki | 15 | — | |
UWDBNTXEKYRMSG
|
7.9 | Ki | 26 | — | |
CRFHZXHUGPCWJA
|
7.9 | IC50 | 8 | — | |
GAROAAIHALTJIR
|
7.9 | IC50 | 3 | Yes | |
HOYCAZAYAZDSGA
|
7.9 | IC50 | 2 | — | |
HTFSQZHIWGSTMP
|
7.9 | IC50 | 2 | — | |
HYCRTUWVJJGNKA
|
7.9 | IC50 | 4 | — | |
JALSZBXKSDMYIN
|
7.9 | IC50 | 2 | — | |
JBKRHKORBCTVLD
|
7.9 | IC50 | 2 | — | |
KBNSMUBNIUALHR
|
7.9 | IC50 | 3 | — | |
MMVLETOTGHDVPQ
|
7.9 | IC50 | 7 | — | |
MVVLRGOQAYKEMN
|
7.9 | IC50 | 2 | — | |
MVVLRGOQAYKEMN
|
7.9 | IC50 | 2 | — |