Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OPVKJVDDNDEKSB
|
8.1 | IC50 | 2 | — | |
DTZJZNAWJBWOKO
|
8.1 | IC50 | 2 | — | |
VGNWKKQVJCEBCJ
|
8.1 | IC50 | 3 | — | |
BKIGTXQKUBIVPY
|
8.1 | IC50 | 2 | — | |
DASFSPDIWCMVRW
|
8.1 | IC50 | 21 | — | |
LPAKCPZPWXQFRB
|
8.1 | IC50 | 2 | — | |
MXPLKNYFRWTHPW
|
8.1 | IC50 | 2 | — | |
NNZRYGISYKGSCW
|
8.1 | IC50 | 3 | — | |
RBMOLIOJAWRTIV
|
8.1 | IC50 | 5 | — | |
SJJYWHYLVWAUQL
|
8.1 | Ki | 2 | — | |
YRIZEPGWRQGUBO
|
8.1 | IC50 | 4 | Yes | |
ZCCJKVBTHCOISJ
|
8.1 | IC50 | 46 | — | |
QWDOEIJNIDENOC
|
8.0 | IC50 | 3 | — | |
BLEFJHDCLNVQNS
|
8.0 | IC50 | 3 | — | |
LMBOMGUIBWYBDA
|
8.0 | IC50 | 3 | — | |
SVDPMUQDJQIHAL
|
8.0 | IC50 | 2 | — | |
AYNBVKYDBZJRNM
|
8.0 | IC50 | 2 | Yes | |
GGIPEVUWPMVPNG
|
8.0 | IC50 | 5 | Yes | |
GRXDRZBYCBQOFV
|
8.0 | IC50 | 2 | — | |
HCBIHPMBVAMDAB
|
8.0 | IC50 | 3 | — | |
OAOPWYXDCLIWEH
|
8.0 | IC50 | 2 | — | |
YNNQCQWREXRBLV
|
8.0 | IC50 | 2 | — | |
BFSNADDVVFYGDC
|
8.0 | IC50 | 2 | — | |
BNFUMIPEQQICKC
|
8.0 | Ki | 2 | — | |
BOWYXGHFMQMXPT
|
8.0 | Ki | 9 | — | |
CJSJFNXXOCNUIQ
|
8.0 | IC50 | 2 | — | |
FGUXNPZAGDXHPG
|
8.0 | IC50 | 2 | — | |
FQVJSQJPMQVZKV
|
8.0 | IC50 | 3 | Yes | |
GJKVMXDBPDDFHI
|
8.0 | Ki | 27 | — | |
GQLWKGVBOIYMTN
|
8.0 | Ki | 35 | — | |
GWMLTDIKRRDXOE
|
8.0 | IC50 | 3 | Yes | |
GXJSLIOOPZRPEV
|
8.0 | Ki | 34 | — | |
HOPYTUITHBXQSC
|
8.0 | IC50 | 5 | Yes | |
HPJPZVODQVTPBB
|
8.0 | IC50 | 3 | — | |
IOBVCHJTLVPPBR
|
8.0 | Ki | 39 | — | |
JAHZZERYOWPURL
|
8.0 | IC50 | 3 | — | |
KLJHWMRQVFONEN
|
8.0 | Ki | 2 | — | |
KRIUNPBAQZGFQA
|
8.0 | Ki | 76 | — | |
LFDJFILTWUNEEP
|
8.0 | IC50 | 6 | Yes | |
LYNBNVBMAGDJRW
|
8.0 | Ki | 81 | — | |
MFMXAWQGPQXDRJ
|
8.0 | Ki | 27 | — | |
NCBGQRJCNZUAKT
|
8.0 | IC50 | 3 | Yes | |
SEVCBWKJSOLMNQ
|
8.0 | Ki | 38 | — | |
VPEYPVPNDMIFEL
|
8.0 | IC50 | 3 | — | |
WBAWCNRBKDEMDU
|
8.0 | Ki | 2 | — | |
ZHJBAEFYMAHRNP
|
8.0 | Ki | 2 | — | |
ZRTDVTOMXDEXHC
|
8.0 | IC50 | 2 | — | |
JYVCLVPNSVUQHC
|
8.0 | IC50 | 2 | — | |
MXYMWTPPSBKBGN
|
8.0 | IC50 | 2 | — | |
ZIZAJYWIUBTSRC
|
8.0 | IC50 | 2 | — |