Target Details
| UniProt AC | Q96GD4 |
|---|---|
| Gene Symbol | AURKB |
| Protein Name | Aurora kinase B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,030
- Clinical molecules 351
- Avg pChEMBL 7.32
KEGG Pathways (2)
Active Molecules (2,030)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QTTGVGLTCILDCA
|
11.0 | Kd | 7 | — | |
IALDYVNFZAPNJV
|
10.9 | Kd | 11 | — | |
CWBIOTBDHJUHCV
|
10.4 | IC50 | 3 | — | |
SNBMLCRFYZAAAX
|
10.3 | IC50 | 3 | — | |
PUFIZMIVJDQOHA
|
10.3 | IC50 | 3 | — | |
LHDWVUBCEIVHFK
|
10.2 | IC50 | 2 | — | |
RWDHVFTXNBLJFJ
|
10.2 | IC50 | 2 | — | |
QJMIUPZFDRLJHJ
|
10.1 | IC50 | 2 | — | |
NNQHKTWARZSGTQ
|
10.0 | Kd | 7 | — | |
PSYMLFSTUXAGFZ
|
9.8 | IC50 | 3 | — | |
BPXZXMRLFSWKLW
|
9.7 | IC50 | 3 | — | |
NHLHBOLWWGNMJH
|
9.7 | IC50 | 2 | — | |
BNTYNTVACAGJNE
|
9.7 | IC50 | 2 | — | |
WUTICGGSWNCYCY
|
9.7 | IC50 | 2 | — | |
ITKXNAMPORNHCX
|
9.7 | IC50 | 2 | — | |
ORMLOSONIQIDBI
|
9.6 | IC50 | 3 | — | |
DHNWCWGJFSTRBB
|
9.6 | IC50 | 3 | — | |
GZBZDQBLAIACNB
|
9.6 | IC50 | 3 | — | |
TUVCZMWCKOCSGF
|
9.6 | IC50 | 3 | — | |
GBKAFRSEJQCGNT
|
9.5 | IC50 | 2 | — | |
ZYCYNVIAJAEECH
|
9.5 | IC50 | 2 | — | |
BBNMVNJADAIHAK
|
9.5 | IC50 | 2 | — | |
VSIZGIFPGSTFOV
|
9.5 | IC50 | 3 | — | |
KPFKWRJCTOGYCX
|
9.5 | IC50 | 2 | — | |
CGDYRZUPKPBLND
|
9.5 | IC50 | 2 | — | |
JMHMGIHHTONCMK
|
9.5 | IC50 | 3 | — | |
JMSLGFQQYRJYBH
|
9.5 | IC50 | 2 | — | |
KMFBAJNOTSSVEC
|
9.5 | IC50 | 2 | — | |
UXYIPHKBTFKDMP
|
9.5 | IC50 | 3 | — | |
VSUHZFYKALKPLP
|
9.5 | IC50 | 2 | — | |
JWSHIVZYYNSBPC
|
9.5 | IC50 | 3 | — | |
LJMKRAKDJVPMIO
|
9.5 | IC50 | 3 | — | |
YGQJBWJOHRVWHU
|
9.5 | IC50 | 3 | — | |
GBJVVSCPOBPEIT
|
9.4 | IC50 | 13 | Yes | |
IHDFFGIONOKCLR
|
9.4 | IC50 | 3 | — | |
UFVBHPSYTMXORI
|
9.4 | IC50 | 2 | — | |
XZHGTQKZIVZJHA
|
9.4 | IC50 | 2 | — | |
HEBODLJXGULWNN
|
9.4 | IC50 | 3 | — | |
LSOZVYDETZGJRK
|
9.4 | IC50 | 3 | — | |
NKKNQMFHKZEGQU
|
9.4 | IC50 | 5 | — | |
SICPNVSSMIOAEC
|
9.4 | IC50 | 3 | — | |
WACBDIUIBDYGCE
|
9.4 | IC50 | 3 | — | |
YNPQIFHMRSVLHW
|
9.4 | IC50 | 3 | — | |
FWHSZSDGPFVMOC
|
9.3 | IC50 | 3 | — | |
IWBOFXHEGIMYAM
|
9.3 | IC50 | 3 | — | |
RKZPJUYYKFXMLU
|
9.3 | IC50 | 3 | — | |
LHVUZIHFLUPGOR
|
9.3 | Ki | 3 | — | |
MZNBFJHMZMXTSD
|
9.3 | IC50 | 3 | — | |
NVWZWRFWZNYFRS
|
9.3 | IC50 | 2 | — | |
PGGKNOUMRNIDKJ
|
9.3 | IC50 | 2 | — |