Target Details
| UniProt AC | Q96D31 |
|---|---|
| Gene Symbol | ORAI1 |
| Protein Name | Calcium release-activated calcium channel protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07856 (Orai-1) |
Summary
- Multi-target molecules 97
- Clinical molecules 0
- Avg pChEMBL 6.66
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (97)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MPBVNNVYYBZUBT
|
7.7 | IC50 | 2 | — | |
VEEFSWBIYMHIDZ
|
7.7 | IC50 | 2 | — | |
NETRIIZSLUUEKM
|
7.6 | IC50 | 2 | — | |
UAQNSPWVOORBLB
|
7.5 | IC50 | 2 | — | |
KFLALJIMRGRRSE
|
7.5 | IC50 | 2 | — | |
GHVJBFUZYPACNM
|
7.5 | IC50 | 2 | — | |
XKCPTMMOWPCFIC
|
7.4 | IC50 | 2 | — | |
VZMFKIDZMKHSBA
|
7.4 | IC50 | 2 | — | |
OBECWQKEMCDNIH
|
7.3 | IC50 | 2 | — | |
HACUWFNZXMLECQ
|
7.3 | IC50 | 2 | — | |
MYWRMJZQVRBGIM
|
7.3 | IC50 | 2 | — | |
XCTONGNRTZPQBT
|
7.3 | IC50 | 2 | — | |
LUIVHTZNEFYWML
|
7.3 | IC50 | 2 | — | |
AXWNMOKUOCPKID
|
7.3 | IC50 | 2 | — | |
RQQJJXVETXFINY
|
7.3 | Ki | 5 | — | |
UILDQRFIEXOIGD
|
7.2 | IC50 | 2 | — | |
UOXHLYMLCPPNGX
|
7.2 | IC50 | 2 | — | |
CWFWVONQCHIWTH
|
7.2 | IC50 | 2 | — | |
DUFHAWGLGXXRBG
|
7.2 | IC50 | 2 | — | |
JLGFZBLOESSPHG
|
7.2 | IC50 | 2 | — | |
VFULESSGOQEDRW
|
7.2 | IC50 | 2 | — | |
WVXWEWXVLIUSCI
|
7.2 | IC50 | 2 | — | |
CEEWGQSGRMFCET
|
7.1 | IC50 | 2 | — | |
NYDXXCFKGFJZIR
|
7.1 | IC50 | 2 | — | |
ZKAHFFVNALZECX
|
7.1 | IC50 | 4 | — | |
LXBHQPCJVRNUPD
|
7.1 | IC50 | 2 | — | |
DRJYDHRCHDJURL
|
7.0 | IC50 | 2 | — | |
BEBHBILBEVKHHU
|
7.0 | IC50 | 2 | — | |
FWFALJHSGGWRGC
|
6.9 | IC50 | 2 | — | |
QQMKTHUGOQDEIL
|
6.9 | IC50 | 3 | — | |
LCFBZFUUCYXAAS
|
6.9 | IC50 | 2 | — | |
SYEBDSIZVIIHNS
|
6.9 | IC50 | 2 | — | |
SNKYIAUGZGHVTO
|
6.9 | IC50 | 2 | — | |
XSLDNIVHKPCLEH
|
6.8 | IC50 | 2 | — | |
FQBXOFLHBKDTPO
|
6.8 | IC50 | 2 | — | |
RSATXOOGPNSIBY
|
6.8 | IC50 | 2 | — | |
FECPMVWBSZDHPR
|
6.8 | IC50 | 2 | — | |
OYBILUBTBUJCSL
|
6.8 | IC50 | 2 | — | |
ZZXATCCXNXZJSE
|
6.8 | IC50 | 2 | — | |
AFWWKCQISQJWEL
|
6.7 | IC50 | 2 | — | |
RFTNCPFRYIPUHX
|
6.7 | IC50 | 2 | — | |
CJSSCSFJKBMVPA
|
6.7 | IC50 | 2 | — | |
KOAUWBDKSVKMMA
|
6.7 | IC50 | 2 | — | |
OYSZVMLSJODPRA
|
6.7 | IC50 | 2 | — | |
OINQZFVFJYCDQI
|
6.7 | IC50 | 2 | — | |
MOXHODGYJMWHOR
|
6.7 | IC50 | 2 | — | |
GFEIWXNLDKUWIK
|
6.6 | IC50 | 2 | — | |
AVNNWXCNOLKWDE
|
6.6 | IC50 | 2 | — | |
ZGOGOEHAPKNVDW
|
6.6 | IC50 | 2 | — | |
GFXQZHGZXMQDCU
|
6.6 | IC50 | 2 | — |