Target Details
| UniProt AC | Q96BR1 |
|---|---|
| Gene Symbol | SGK3 |
| Protein Name | Serine/threonine-protein kinase Sgk3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) PF00787 (PX) |
Summary
- Multi-target molecules 16
- Clinical molecules 4
- Avg pChEMBL 6.62
KEGG Pathways (2)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
IIRWNGPLJQXWFJ
|
7.3 | IC50 | 21 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
YYLKKYCXAOBSRM
|
7.0 | Kd | 191 | — | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
VYIKAHZTFTUSJO
|
6.7 | IC50 | 3 | — | |
WINHZLLDWRZWRT
|
6.7 | Kd | 201 | Yes | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
RTFQFPZKDYMMMJ
|
6.5 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
PIQCTGMSNWUMAF
|
6.0 | Kd | 137 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
XZXHXSATPCNXJR
|
6.0 | Kd | 165 | Yes |