Target Details
| UniProt AC | Q96BI3 |
|---|---|
| Gene Symbol | APH1A |
| Protein Name | Gamma-secretase subunit APH-1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF06105 (Aph-1) |
Summary
- Multi-target molecules 1,927
- Clinical molecules 1
- Avg pChEMBL 7.37
KEGG Pathways (3)
Active Molecules (1,927)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OFTOYMCRCCAFGE
|
9.4 | IC50 | 6 | — | |
YXESTJAWJQYHFN
|
9.4 | IC50 | 6 | — | |
ULSSJYNJIZWPSB
|
9.4 | IC50 | 7 | — | |
BPRBCTZEWQCYNJ
|
9.4 | IC50 | 6 | — | |
FFKAEWHVIHHSLK
|
9.4 | IC50 | 6 | — | |
CAYZCIFYSFVVTI
|
9.4 | IC50 | 6 | — | |
FEIXZFKKQUZLPW
|
9.4 | IC50 | 6 | — | |
KIKHYLCLMBUGBG
|
9.4 | IC50 | 6 | — | |
XXTPLLFHAQMCTN
|
9.4 | IC50 | 6 | — | |
YCBAQKQAINQRFW
|
9.4 | IC50 | 6 | — | |
JAYWWVGRDYLXQP
|
9.4 | IC50 | 6 | — | |
LBJYPLZODCWHKE
|
9.4 | IC50 | 6 | — | |
MAZVAJBBINZFPI
|
9.4 | IC50 | 6 | — | |
RGYAICMEYBJRDC
|
9.4 | IC50 | 6 | — | |
GVVYZJLUZCRFEO
|
9.4 | IC50 | 6 | — | |
DJJNHFXUJZZRIH
|
9.3 | IC50 | 6 | — | |
KPILYJMXAJUQSK
|
9.3 | IC50 | 6 | — | |
VONONKABRHIFEM
|
9.3 | IC50 | 6 | — | |
POIOTSUEZZWFIU
|
9.3 | IC50 | 6 | — | |
IYOICEQASLKVSF
|
9.3 | IC50 | 6 | — | |
OQUHWHUICWTGQJ
|
9.3 | IC50 | 6 | — | |
XVYHWQOGORTPLY
|
9.3 | IC50 | 6 | — | |
FFHJMTQXXIYCKU
|
9.3 | IC50 | 6 | — | |
TYYKLJZPSLNJOH
|
9.3 | IC50 | 6 | — | |
VUDMLJPTMCGJLN
|
9.3 | IC50 | 6 | — | |
WFWGAWVCMNUSPE
|
9.3 | IC50 | 6 | — | |
IWPLJEVPDSNRHR
|
9.3 | IC50 | 6 | — | |
YZUZOPGLOYYWKD
|
9.3 | IC50 | 6 | — | |
ZWYBSWYYUMKRPV
|
9.3 | IC50 | 6 | — | |
XSHZFWXNHJNUBT
|
9.3 | IC50 | 6 | — | |
YAEBTEGCKUXQCL
|
9.2 | IC50 | 6 | — | |
YMCMJVOZVFFIKZ
|
9.2 | IC50 | 6 | — | |
ZZGIOVGHNKXQNY
|
9.2 | IC50 | 6 | — | |
OTXHDBQTORDBPA
|
9.2 | IC50 | 6 | — | |
IACJSTAPBNKIAR
|
9.2 | IC50 | 6 | — | |
LWOBGHMKQHIENT
|
9.2 | IC50 | 6 | — | |
HKLRXCRZQQZDET
|
9.2 | IC50 | 6 | — | |
IHTDUZYFQXWLFI
|
9.2 | IC50 | 6 | — | |
KLJYBGHIYLAIJK
|
9.2 | IC50 | 6 | — | |
NAQPWAVBAAJHPY
|
9.2 | IC50 | 6 | — | |
VEHFINFYUNHULM
|
9.2 | IC50 | 6 | — | |
CEOHFPLVFGSEBG
|
9.2 | IC50 | 6 | — | |
FJLCFJOFTFRWRX
|
9.2 | IC50 | 6 | — | |
MKHGYZOIWHXDGL
|
9.2 | IC50 | 6 | — | |
VJTZQYXICDNCMU
|
9.2 | IC50 | 6 | — | |
MCOGETVHCTZXCD
|
9.1 | IC50 | 6 | — | |
BAPPJDHHRPNBPT
|
9.1 | IC50 | 6 | — | |
IMLZVQJYFBAVIP
|
9.1 | IC50 | 6 | — | |
PAYDYCBYWDPAKX
|
9.1 | IC50 | 6 | — | |
VWPBQGYFODMQHR
|
9.1 | IC50 | 6 | — |