Target Details
| UniProt AC | Q96BI3 |
|---|---|
| Gene Symbol | APH1A |
| Protein Name | Gamma-secretase subunit APH-1A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF06105 (Aph-1) |
Summary
- Multi-target molecules 1,927
- Clinical molecules 1
- Avg pChEMBL 7.37
KEGG Pathways (3)
Active Molecules (1,927)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLPZMVARYYWCLF
|
7.5 | IC50 | 6 | — | |
UTKNCPXIXJKKPY
|
7.5 | IC50 | 6 | — | |
ZALNMHMJXFINHH
|
7.5 | IC50 | 6 | — | |
DLMNHZHQGVMRJB
|
7.5 | IC50 | 6 | — | |
NDVMOVOEROCRIO
|
7.5 | IC50 | 6 | — | |
RJBHTARGFMGGBA
|
7.5 | IC50 | 6 | — | |
XJKKUMGGCRZLGE
|
7.5 | IC50 | 6 | — | |
XKKPUSBAPFUJJA
|
7.5 | IC50 | 6 | — | |
XYQDAYZDRBKPNR
|
7.5 | IC50 | 6 | — | |
ZLEUKGZKAVGDKU
|
7.5 | IC50 | 6 | — | |
ZRCZGEIHIFDAPM
|
7.5 | IC50 | 6 | — | |
CXJQWJBRXYDTFP
|
7.5 | IC50 | 6 | — | |
DDVQYGCPVJHCFB
|
7.5 | IC50 | 6 | — | |
GZGVHQMYSJNKMG
|
7.5 | IC50 | 6 | — | |
IFBOJVNFJCLRIC
|
7.5 | IC50 | 6 | — | |
JEBOHMDITPRILC
|
7.5 | IC50 | 6 | — | |
KKFRXIHTRCQMHV
|
7.5 | IC50 | 7 | — | |
SUYIHEGPYVNQBO
|
7.5 | IC50 | 6 | — | |
WGSSDSCDGURRHH
|
7.5 | IC50 | 7 | — | |
XRFPNOICOXIYQT
|
7.5 | IC50 | 6 | — | |
GPJQZPLKOWGOSM
|
7.5 | IC50 | 6 | — | |
LFZXHYJFDCRIGT
|
7.5 | IC50 | 6 | — | |
LFZXHYJFDCRIGT
|
7.5 | IC50 | 6 | — | |
LPLQFQASZSTOMW
|
7.5 | IC50 | 6 | — | |
NXPQBVTVDAZRRT
|
7.5 | IC50 | 6 | — | |
WQCCBXNMIRUREM
|
7.5 | IC50 | 6 | — | |
YTBSSZLYKCFJCT
|
7.5 | IC50 | 6 | — | |
HGUUOHWKCPBRDE
|
7.5 | IC50 | 6 | — | |
IQTCDSQBHHTVBN
|
7.5 | IC50 | 6 | — | |
NNOFJBXUZPTMFY
|
7.5 | IC50 | 6 | — | |
ODEIUBHPOCSQNG
|
7.5 | IC50 | 6 | — | |
SJGAOAJELVBEMC
|
7.5 | IC50 | 6 | — | |
SOWUEDNFEKMNJN
|
7.5 | IC50 | 6 | — | |
UVFIJTYAZWJSFV
|
7.5 | IC50 | 6 | — | |
VOAVANGLSKPOPN
|
7.5 | IC50 | 6 | — | |
WJWXNUKTBZWHEM
|
7.5 | IC50 | 6 | — | |
ZHNDWSFRNPTACV
|
7.5 | IC50 | 7 | — | |
KRXBKHKDFUKPLA
|
7.5 | IC50 | 6 | — | |
LBRVZRHWWSHEBP
|
7.5 | IC50 | 6 | — | |
AOISQQKLSIPOKV
|
7.4 | IC50 | 6 | — | |
HJZVCQVBPMDUMS
|
7.4 | IC50 | 7 | — | |
JNSRRQZTTJNISW
|
7.4 | IC50 | 6 | — | |
KBBNHQZMJPGKNW
|
7.4 | IC50 | 6 | — | |
KGZQTRVMNLJDEO
|
7.4 | IC50 | 6 | — | |
KOSXCVWYEAFBIP
|
7.4 | IC50 | 6 | — | |
KXRFLRBMOABABP
|
7.4 | IC50 | 6 | — | |
MURCDOXDAHPNRQ
|
7.4 | IC50 | 8 | — | |
MVLQSAIIKQCXDH
|
7.4 | IC50 | 6 | — | |
NUAQUNTYWPZJMU
|
7.4 | Ki | 6 | — | |
XAGIJOHXUNDGDQ
|
7.4 | IC50 | 6 | — |