Target Details
| UniProt AC | Q969S8 |
|---|---|
| Gene Symbol | HDAC10 |
| Protein Name | Polyamine deacetylase HDAC10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 1,942
- Clinical molecules 427
- Avg pChEMBL 7.06
KEGG Pathways (3)
Active Molecules (1,942)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LAMIXXKAWNLXOC
|
7.8 | IC50 | 12 | Yes | |
NJTBXOKFMYGINE
|
7.8 | IC50 | 11 | — | |
NXGMKXAFBYEHBZ
|
7.8 | IC50 | 7 | Yes | |
SKTBGPXTJPTFJR
|
7.8 | IC50 | 11 | — | |
UHPVVZUVOPNTDE
|
7.8 | IC50 | 12 | — | |
ULIOZFPEJTVCBT
|
7.8 | IC50 | 11 | — | |
YMLSAIDCGOYCCA
|
7.8 | IC50 | 11 | — | |
FUUWQMNGOYFALL
|
7.8 | IC50 | 11 | — | |
KYMAKPZTKUPPRK
|
7.8 | IC50 | 11 | — | |
SGTCWQOXXQUYHN
|
7.8 | IC50 | 6 | Yes | |
DQIMPFMQPBIJFZ
|
7.8 | IC50 | 11 | — | |
HOPNPVAERWNDPG
|
7.8 | IC50 | 11 | — | |
NJEYLEUCEPGDMG
|
7.8 | IC50 | 11 | — | |
RKGDKTNUCYVAEK
|
7.8 | IC50 | 11 | — | |
ZTLUHMBJQIQLKN
|
7.8 | IC50 | 12 | — | |
BYKMCJLDXBMWTO
|
7.8 | IC50 | 7 | Yes | |
IJSZCGGEDBEPHU
|
7.8 | IC50 | 11 | — | |
ZPAHLBXHWVNFMV
|
7.8 | IC50 | 15 | — | |
GYWQCXUVPDWXRB
|
7.8 | IC50 | 11 | — | |
HRMYEEYQEBQZKK
|
7.8 | IC50 | 11 | — | |
HWXIALUKOFRCLZ
|
7.8 | IC50 | 12 | — | |
ICZBBQCOKLJCOL
|
7.8 | IC50 | 11 | — | |
IKSWFKPGSLOVSP
|
7.8 | IC50 | 12 | — | |
OFRPIMCNWXHVHW
|
7.8 | IC50 | 11 | — | |
QJNQAMKQPQVGHL
|
7.8 | IC50 | 5 | — | |
RUSJYWZWAOCFFO
|
7.8 | IC50 | 7 | Yes | |
UHFLTFWSPYVZHA
|
7.8 | IC50 | 11 | — | |
VZFNPGQXAMLZHT
|
7.8 | IC50 | 11 | — | |
XVEOCYHWWWIAJH
|
7.8 | IC50 | 11 | — | |
ZHYWBQIDWBAPRN
|
7.8 | IC50 | 11 | — | |
YKOJCIKYDZHWDT
|
7.7 | Ki | 12 | Yes | |
QWAGLXWBHCFGBD
|
7.7 | IC50 | 6 | Yes | |
GNPOWSZXVBHRHU
|
7.7 | IC50 | 11 | — | |
HRKITJYWVNASHR
|
7.7 | Ki | 12 | Yes | |
IKVGYSSTVXNKDM
|
7.7 | IC50 | 11 | — | |
JHDKZFFAIZKUCU
|
7.7 | Ki | 11 | — | |
MZTDGAQDNCVZMT
|
7.7 | IC50 | 11 | — | |
RCDIZKAYZBEALO
|
7.7 | Ki | 11 | Yes | |
RDNBSSIISDHNPJ
|
7.7 | IC50 | 11 | — | |
UQIMEFHEVVKGJC
|
7.7 | IC50 | 7 | Yes | |
YRRVLBINSXVLFM
|
7.7 | IC50 | 12 | — | |
ZCQUIFOQIMJOHM
|
7.7 | IC50 | 11 | Yes | |
ZJQBOUFZLSVUBC
|
7.7 | IC50 | 12 | — | |
AYECQXDGPKKAOJ
|
7.7 | IC50 | 11 | — | |
DMXROUYLQHFRCS
|
7.7 | Ki | 7 | Yes | |
FFQLSSOAWSFFMY
|
7.7 | IC50 | 15 | — | |
ILNZTCJWQPCPCA
|
7.7 | IC50 | 11 | — | |
IUVUZERDURJGCP
|
7.7 | IC50 | 11 | — | |
JITONGQJSJWWMH
|
7.7 | IC50 | 11 | — | |
KASXKFPWIZYBSG
|
7.7 | IC50 | 11 | Yes |