Target Details
| UniProt AC | Q969S8 |
|---|---|
| Gene Symbol | HDAC10 |
| Protein Name | Polyamine deacetylase HDAC10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 1,942
- Clinical molecules 427
- Avg pChEMBL 7.06
KEGG Pathways (3)
Active Molecules (1,942)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NEUFRFUBRUCEHM
|
8.1 | IC50 | 11 | — | |
AZUDZSYTIWKGBN
|
8.1 | IC50 | 11 | — | |
ILCBWDQDWOLKIQ
|
8.1 | IC50 | 7 | — | |
IXKLILPHPNZHNB
|
8.1 | IC50 | 12 | Yes | |
KUEQWBIGMIIMRB
|
8.1 | IC50 | 11 | — | |
LZODJSNRNSCPJV
|
8.1 | IC50 | 7 | — | |
RVWKGSCHYRXCNC
|
8.1 | Ki | 11 | Yes | |
VUHMGFRTADPQOA
|
8.1 | IC50 | 11 | — | |
ZUUNAMZBBZETFV
|
8.1 | IC50 | 11 | — | |
BNXWGPQAXDBKJF
|
8.0 | IC50 | 11 | Yes | |
PDRHOJIVDMXSPA
|
8.0 | IC50 | 3 | — | |
XLYWAZNXULUIKN
|
8.0 | IC50 | 11 | — | |
HUKZXIATPPFLSE
|
8.0 | IC50 | 11 | Yes | |
QXIIXGYKPYLMDY
|
8.0 | IC50 | 11 | — | |
WFODACKMLVBMPT
|
8.0 | IC50 | 11 | — | |
XPQULOSXGAVNNQ
|
8.0 | IC50 | 6 | Yes | |
BDTAPZUZFJRPNM
|
8.0 | IC50 | 12 | Yes | |
FBXQCHJAZBIFFB
|
8.0 | IC50 | 12 | Yes | |
HUFMIDSGMTUTRL
|
8.0 | IC50 | 12 | — | |
IQONMOHAPASEMF
|
8.0 | IC50 | 11 | — | |
JOBWAXWKZPONDF
|
8.0 | IC50 | 11 | — | |
QRASJFWGSXNPPD
|
8.0 | IC50 | 11 | — | |
UYCGYJBWLFVKGB
|
8.0 | IC50 | 12 | Yes | |
VXQMHJZDOMPYKM
|
8.0 | IC50 | 11 | — | |
ZEUHZRVYLQKSEE
|
8.0 | IC50 | 11 | — | |
ZSXALGICOGVKEL
|
8.0 | IC50 | 12 | Yes | |
OJIBZKCCZAUUJU
|
8.0 | IC50 | 11 | — | |
OEDQYVKPPIYBLX
|
8.0 | IC50 | 6 | Yes | |
GAZWXVIVAKKMPK
|
8.0 | IC50 | 6 | — | |
IDXZLMIYGOBMPS
|
8.0 | IC50 | 11 | — | |
ILCBWDQDWOLKIQ
|
8.0 | IC50 | 7 | — | |
NYJOCLMLIASQTH
|
8.0 | IC50 | 7 | — | |
PQSQTRKAQOTEHG
|
8.0 | IC50 | 12 | — | |
VWBBPADKULAZAT
|
8.0 | IC50 | 11 | Yes | |
XVGBJXUAVWXLJX
|
8.0 | IC50 | 8 | — | |
YYSCXBPFYMVUDP
|
8.0 | IC50 | 7 | — | |
YYSCXBPFYMVUDP
|
8.0 | IC50 | 7 | — | |
LJFNWCGSOPRFNA
|
8.0 | IC50 | 12 | Yes | |
NEZCKIVFZVYNMQ
|
8.0 | IC50 | 13 | Yes | |
BGEMMLGLCIAYAX
|
7.9 | IC50 | 11 | — | |
HLYPKXDQBACOJP
|
7.9 | IC50 | 11 | Yes | |
LOWILHBHMVLGAV
|
7.9 | IC50 | 11 | — | |
RQHGHGKQPZXBJW
|
7.9 | IC50 | 11 | — | |
XGUBSOZYNYGGSV
|
7.9 | IC50 | 11 | — | |
RUVXTVKADDBLBK
|
7.9 | IC50 | 11 | — | |
KAFPWADPNJMVFZ
|
7.9 | IC50 | 11 | — | |
AQIOMPMNFDEIJO
|
7.9 | IC50 | 12 | Yes | |
BBLKKBHWHCNSHW
|
7.9 | IC50 | 11 | — | |
DTDNZGWJQYUFBL
|
7.9 | IC50 | 11 | — | |
JPJYOPNEGMWFJL
|
7.9 | IC50 | 15 | Yes |