Target Details
| UniProt AC | Q969S8 |
|---|---|
| Gene Symbol | HDAC10 |
| Protein Name | Polyamine deacetylase HDAC10 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 1,942
- Clinical molecules 427
- Avg pChEMBL 7.06
KEGG Pathways (3)
Active Molecules (1,942)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HVAMCPMMTPHGBZ
|
9.7 | IC50 | 12 | — | |
STYUEVXPOBLDCO
|
9.7 | IC50 | 12 | Yes | |
UCPPLLAVVTUHRE
|
9.7 | IC50 | 14 | Yes | |
VODSDFCUCFMZGN
|
9.7 | IC50 | 14 | Yes | |
VXQMEGLYMWVBHB
|
9.7 | IC50 | 6 | — | |
BCSAECULXJTTAB
|
9.5 | IC50 | 12 | — | |
CCDVRDJZGFEHAS
|
9.5 | IC50 | 14 | Yes | |
GREXOPZRGSQSHE
|
9.5 | IC50 | 11 | — | |
ZIXGFQGSZCYOCA
|
9.5 | IC50 | 11 | — | |
MGSMSINQVPOBFG
|
9.4 | IC50 | 12 | — | |
NXFALCZBQFKESM
|
9.4 | IC50 | 14 | Yes | |
CALHFQHOBJNLIX
|
9.3 | IC50 | 6 | — | |
VEDPEVJAYWVUSJ
|
9.3 | IC50 | 7 | — | |
VEDPEVJAYWVUSJ
|
9.3 | IC50 | 7 | — | |
YPXRCUVTZDXVHY
|
9.2 | IC50 | 7 | — | |
ZGYDQVJYONGOFO
|
9.1 | IC50 | 12 | — | |
TWJZFXHSPBBPNI
|
9.1 | IC50 | 5 | — | |
YNDXKTMBUARZGX
|
9.1 | IC50 | 11 | — | |
PPEIAJKMCSPOIO
|
9.0 | IC50 | 11 | — | |
CSOPQBAMSLNMTB
|
9.0 | IC50 | 12 | Yes | |
IDFCPXHALXHUKZ
|
9.0 | IC50 | 11 | — | |
JTIATMCBWUQBGH
|
9.0 | IC50 | 7 | — | |
NWSVQMVAPKFALM
|
9.0 | IC50 | 12 | Yes | |
OHRURASPPZQGQM
|
9.0 | IC50 | 9 | — | |
OZVBWIKRBIZHCH
|
9.0 | IC50 | 11 | — | |
QWRAOGOVSCMHRF
|
9.0 | IC50 | 11 | — | |
WMMGXRCXFKMSGF
|
9.0 | IC50 | 14 | Yes | |
XJEGEVAGSHPOIG
|
9.0 | IC50 | 11 | — | |
SVPPYXRDCMLVCS
|
9.0 | IC50 | 12 | — | |
JQUGGCHYIXURKK
|
8.9 | IC50 | 11 | — | |
MUIRESFGWICKLJ
|
8.9 | IC50 | 11 | — | |
UOEXMKBLKQPTKA
|
8.9 | IC50 | 12 | Yes | |
WOGPSXAJPRAXBA
|
8.9 | Ki | 8 | — | |
PJNFGPBZRCJQFS
|
8.9 | IC50 | 12 | Yes | |
ABJDGWXKAMVWGP
|
8.8 | IC50 | 7 | — | |
FATABLVXWFWXHK
|
8.8 | IC50 | 12 | Yes | |
CUHDSDLVRCISIT
|
8.8 | IC50 | 11 | — | |
RIHKXPFNMAZMOA
|
8.8 | IC50 | 11 | — | |
WEUZJBFBMQCGSG
|
8.8 | IC50 | 11 | — | |
XCYPPRCLPXVRLG
|
8.8 | IC50 | 11 | — | |
IXTBKGBJNGTKQS
|
8.8 | IC50 | 12 | — | |
JMUDLVWSKDYNSZ
|
8.8 | IC50 | 11 | — | |
AACFFQPNGHLYEG
|
8.7 | IC50 | 11 | — | |
LZEMGHTYCJXNLM
|
8.7 | IC50 | 11 | — | |
RTKIYFITIVXBLE
|
8.7 | IC50 | 11 | — | |
OHRURASPPZQGQM
|
8.7 | IC50 | 14 | — | |
YLQFHROXRNFGMC
|
8.7 | IC50 | 11 | — | |
BHYPIIUJEQHYIP
|
8.7 | IC50 | 14 | Yes | |
DTTIQSUWHKFPML
|
8.7 | IC50 | 7 | — | |
FQWUNUXAOHTLLG
|
8.7 | IC50 | 12 | Yes |