Target Details
| UniProt AC | Q95PM0 |
|---|---|
| Gene Symbol | rhodesain |
| Protein Name | N/A |
| Organism | Trypanosoma brucei rhodesiense |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF12131 (DUF3586) PF08246 (Inhibitor_I29) PF00112 (Peptidase_C1) |
Summary
- Multi-target molecules 157
- Clinical molecules 0
- Avg pChEMBL 7.82
Active Molecules (157)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YCDLIADNLQNFRV
|
7.4 | IC50 | 2 | — | |
VCKVRMZTLPAQME
|
7.4 | Ki | 2 | — | |
KQRXZKZSIDZXHU
|
7.4 | IC50 | 2 | — | |
SWEBEQUEVFYZAA
|
7.3 | Ki | 2 | — | |
UKMQUUMHKOPROJ
|
7.3 | Ki | 2 | — | |
WJQYKRIBWNZUHM
|
7.3 | IC50 | 2 | — | |
WJQYKRIBWNZUHM
|
7.3 | IC50 | 2 | — | |
AZDILRCJGPIBEA
|
7.3 | Ki | 2 | — | |
IAJKNEKSFREFIT
|
7.3 | Ki | 2 | — | |
SRNVIXNTQNQATR
|
7.3 | Ki | 2 | — | |
VBHYQAVSSHIJNV
|
7.2 | Ki | 3 | — | |
OAIPJBOHJDECBD
|
7.2 | Ki | 2 | — | |
DIOJIFYCWQBZFF
|
7.2 | IC50 | 2 | — | |
DIOJIFYCWQBZFF
|
7.2 | IC50 | 2 | — | |
ZFWBXQAVLYJGIL
|
7.2 | IC50 | 2 | — | |
ZFWBXQAVLYJGIL
|
7.2 | IC50 | 2 | — | |
VJNSFGVHSJHQMY
|
7.2 | Ki | 2 | — | |
FIJYOQYJGIYCIK
|
7.2 | IC50 | 2 | — | |
FIJYOQYJGIYCIK
|
7.2 | IC50 | 2 | — | |
LHAZNXGFJOVNSB
|
7.2 | Ki | 2 | — | |
NOWCNBDPTWLOJL
|
7.1 | IC50 | 2 | — | |
NOWCNBDPTWLOJL
|
7.1 | IC50 | 2 | — | |
YLRYZOGPSPNUJU
|
7.1 | Ki | 2 | — | |
VXWORSGAIFVSON
|
7.0 | IC50 | 2 | — | |
VXWORSGAIFVSON
|
7.0 | IC50 | 2 | — | |
YTWAAFXYVRVTTR
|
7.0 | Ki | 2 | — | |
ILDMHYFHSBBUCU
|
7.0 | IC50 | 2 | — | |
DXLLSNZJTDGBRA
|
7.0 | IC50 | 4 | — | |
RVTBBZNNLYWUCX
|
7.0 | IC50 | 2 | — | |
RVTBBZNNLYWUCX
|
7.0 | IC50 | 2 | — | |
NHGHQGULMGPVNX
|
6.9 | Ki | 2 | — | |
SKVFLJGZAOSWLB
|
6.9 | Ki | 2 | — | |
JRFCJBAMIBGKTB
|
6.8 | IC50 | 4 | — | |
MEBPGJFXXVRICE
|
6.8 | IC50 | 4 | — | |
DSMGEPBRPIEQKD
|
6.8 | IC50 | 4 | — | |
DSMGEPBRPIEQKD
|
6.8 | IC50 | 3 | — | |
WBIKZQWGHHXZTG
|
6.6 | IC50 | 2 | — | |
WBIKZQWGHHXZTG
|
6.6 | IC50 | 2 | — | |
ROQSYDCGYWIBSQ
|
6.6 | IC50 | 2 | — | |
UVIIBPXEFXJQAV
|
6.6 | Ki | 2 | — | |
BFJRLYQUSWBFAL
|
6.6 | IC50 | 2 | — | |
ILDMHYFHSBBUCU
|
6.5 | IC50 | 2 | — | |
YPTSSADHYSRSLH
|
6.5 | Ki | 2 | — | |
JZEFKJPYPCBZGF
|
6.5 | IC50 | 2 | — | |
XEUCGJSDYZAWTF
|
6.4 | IC50 | 2 | — | |
FTOKQFDENATBOZ
|
6.3 | IC50 | 2 | — | |
PNAOPWGEIDEZMT
|
6.3 | IC50 | 2 | — | |
XFYWHOCFLQPKMK
|
6.3 | Ki | 3 | — | |
YJYSHOADPNSQGD
|
6.2 | IC50 | 4 | — | |
BILXHJBONVDEDN
|
6.2 | IC50 | 2 | — |