Target Details
| UniProt AC | Q92993 |
|---|---|
| Gene Symbol | KAT5 |
| Protein Name | Histone acetyltransferase KAT5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01853 (MOZ_SAS) PF11717 (Tudor-knot) PF17772 (zf-MYST) |
Summary
- Multi-target molecules 131
- Clinical molecules 0
- Avg pChEMBL 6.74
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (131)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JUSFZIPJDUHEMM
|
6.3 | IC50 | 4 | — | |
HRHWETKYVSXITG
|
6.3 | Ki | 2 | — | |
MRWSPFBTCMRIKG
|
6.3 | Ki | 2 | — | |
ZMXHKKITBJLUKM
|
6.3 | Ki | 5 | — | |
OQPGTPAVCKIJGA
|
6.3 | Ki | 2 | — | |
HSFJEZDNBIVIBA
|
6.2 | Ki | 2 | — | |
JWLAJDZKVPQHDN
|
6.2 | Ki | 2 | — | |
OSAPKUVOJCRXOX
|
6.2 | IC50 | 3 | — | |
KWEJMMAITZKAMQ
|
6.2 | Ki | 3 | — | |
VNSQFPFWUAZOTQ
|
6.2 | Ki | 5 | — | |
VQHLTODGZJHRRL
|
6.2 | Ki | 2 | — | |
ABUOWWFPDMGIHU
|
6.2 | Ki | 2 | — | |
FGBITSJINQIUCA
|
6.2 | Ki | 3 | — | |
RZWDESKLSMUQIH
|
6.2 | Ki | 2 | — | |
CSSILMYXWDKRGS
|
6.2 | Ki | 2 | — | |
PCMNWUTUSXYIRT
|
6.2 | IC50 | 3 | — | |
WWFRXLVYYYMFTR
|
6.2 | Ki | 2 | — | |
QYKFOIQECSQWDW
|
6.2 | Ki | 4 | — | |
QRJOXGIEJMPGGH
|
6.1 | Ki | 2 | — | |
FMCCVBHKJSIJEX
|
6.1 | Ki | 4 | — | |
DQUMBPJNDFPLFG
|
6.1 | Ki | 2 | — | |
KFANPTBFAFROHQ
|
6.1 | IC50 | 3 | — | |
NAYMRTIEIIVLHD
|
6.1 | Ki | 5 | — | |
JULSZUGQINBKBM
|
6.1 | Ki | 4 | — | |
YVAODNUHZXTILD
|
6.1 | Ki | 2 | — | |
FNGSGKICDYSQAK
|
6.1 | Ki | 2 | — | |
OPXGFZIMRMXCJW
|
6.1 | Ki | 2 | — | |
UACCCSHYCUCJFW
|
6.1 | IC50 | 3 | — | |
AZJGHRWSOCLSSE
|
6.0 | Ki | 4 | — | |
OBLBXCVBYBHIOD
|
6.0 | Ki | 3 | — | |
YEUSVVVKGKGBGT
|
6.0 | Ki | 3 | — |