Target Details
UniProt ACQ92993
Gene SymbolKAT5
Protein NameHistone acetyltransferase KAT5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF01853 (MOZ_SAS) PF11717 (Tudor-knot) PF17772 (zf-MYST)
Summary
  • Multi-target molecules 131
  • Clinical molecules 0
  • Avg pChEMBL 6.74
Top Co-occurrence Targets
Active Molecules (131)
InChIKey pChEMBL Type Targets Clinical
NRVQEVZNUYQLAS 9.0 Ki 2
NRVQEVZNUYQLAS 8.2 Ki 3
JOFCULIXSWEGCQ 8.1 Ki 3
DTEFNSUWEUOSFX 7.9 Ki 3
PMIUIWMKYCWCIT 7.9 Ki 3
MGRAVCNYGINSME 7.8 Ki 3
VFVZUNDCETVFCY 7.7 Ki 3
GMKQZYDHJJZSBW 7.7 Ki 3
ZGIHMCPGMLLKRH 7.7 Ki 2
DBCRXQGJTHCJJT 7.6 Ki 3
FJZZQNZXTDELJD 7.6 Ki 3
HBKXBYMYQVIYLS 7.5 Ki 3
OIJIORLVSSKPSQ 7.5 Ki 3
SQWYGFRGZFDHCZ 7.5 Ki 3
ZZPPYTBSGIXYHR 7.5 Ki 3
QHPGWXWCBSRYEK 7.4 Ki 2
OTJDPASOKCKBRE 7.3 Ki 3
YNZFMGZYFHYWNM 7.3 Ki 3
HEALUYMIMKNEIO 7.3 Ki 2
ZSKUNGCPEFTJAX 7.3 Ki 3
ZYVLPZNPYZYZES 7.3 Ki 3
DGCCTCIEIMJSQY 7.3 Ki 2
BOIRGEFIRRTNRA 7.2 Ki 2
WYQYLWDBDPTRJH 7.2 Ki 3
KQVDJORREHTNIY 7.2 Ki 2
ZTCKXRDPZQPUAT 7.2 Ki 5
QSIIAMZHCULDGC 7.1 Ki 3
PAOPEAZNZFFYMP 7.1 Ki 2
SIRYYQDQHJOVTK 7.1 Ki 2
GFECGYRHVFAGJS 7.0 Ki 2
JQXCDWCEWHHCOB 7.0 Ki 2
FJVBTCIMEBNXAJ 7.0 Ki 2
URYQEFLKISCQTP 7.0 Ki 2
DQPCLHVPTYVZIU 7.0 Ki 2
MGRAVCNYGINSME 7.0 Ki 2
MXTXGYHNGUAAEW 7.0 Ki 2
SHWIJWSQRJWWBT 7.0 IC50 3
QYEKEYZNXBRTSL 7.0 Ki 5
LXWNJBBICBJZBB 6.9 Ki 3
UQVZRXUOUOWVGZ 6.9 Ki 5
HNHUSASLBMDEED 6.9 Ki 5
RMWMMIJTOPTGGV 6.9 Ki 2
SIUBXLZGASDVQE 6.9 Ki 3
QJQWOQQSEONHLW 6.9 Ki 3
QAQMDGMWXOHYCA 6.8 Ki 2
YDGHDWBDQICHPI 6.8 IC50 3
YJJDAMOMUXHDFT 6.8 IC50 4
FKKPYHKOEUJLJA 6.8 Ki 4
JHHNQSUGVIGBFC 6.8 Ki 5
SIUBXLZGASDVQE 6.8 Ki 3
2D structure