Target Details
| UniProt AC | Q92934 |
|---|---|
| Gene Symbol | BAD |
| Protein Name | Bcl2-associated agonist of cell death |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF10514 (Bcl-2_BAD) |
Summary
- Multi-target molecules 27
- Clinical molecules 0
- Avg pChEMBL 6.72
KEGG Pathways (43)
- Acute myeloid leukemia
- Alzheimer disease
- Amyotrophic lateral sclerosis
- Apoptosis
- Autophagy - animal
- Chemical carcinogenesis - reactive oxygen species
- Chemical carcinogenesis - receptor activation
- Chemokine signaling pathway
- Chronic myeloid leukemia
- Colorectal cancer
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Hepatitis B
- Hepatitis C
- Hepatocellular carcinoma
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- Insulin signaling pathway
- Lipid and atherosclerosis
- Measles
- Melanoma
- Neurotrophin signaling pathway
- Non-small cell lung cancer
- PI3K-Akt signaling pathway
- Pancreatic cancer
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Platinum drug resistance
- Prion disease
- Prostate cancer
- Ras signaling pathway
- Renal cell carcinoma
- Thyroid hormone signaling pathway
- Toxoplasmosis
- Tuberculosis
- VEGF signaling pathway
- Viral carcinogenesis
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (27)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HPLNQCPCUACXLM
|
9.2 | Ki | 11 | — | |
AVHUOMOOFURFSR
|
7.3 | Kd | 2 | — | |
DREKSGOBSPWACW
|
7.3 | IC50 | 2 | — | |
HDMMUGXXXGBXHN
|
7.3 | Kd | 2 | — | |
JLYAXFNOILIKPP
|
7.3 | Kd | 7 | — | |
LKYTZFLMLJYBMS
|
7.3 | Kd | 3 | — | |
LQBVNQSMGBZMKD
|
7.3 | IC50 | 4 | — | |
UZTDMIJOSGYESW
|
7.3 | Kd | 2 | — | |
YTAAEVBCUIZEOM
|
7.3 | Kd | 2 | — | |
ZAXCMHZZKISMCD
|
7.0 | Ki | 2 | — | |
MWJSZKBWGOIWJG
|
6.7 | IC50 | 2 | — | |
DEWYCLMCITZZFP
|
6.6 | Ki | 2 | — | |
NCLFJOPXKSMXQY
|
6.6 | IC50 | 2 | — | |
UGIRPCIVVCEJFA
|
6.6 | Ki | 2 | — | |
WJTXUCODNSFWJQ
|
6.5 | Ki | 2 | — | |
BXXWCEVDYNCKIB
|
6.4 | Ki | 2 | — | |
YOALHDWNEMCDAJ
|
6.4 | IC50 | 2 | — | |
KGDQVKRMGYAUAI
|
6.3 | Ki | 2 | — | |
XRQBYGKJAKJADI
|
6.3 | Ki | 2 | — | |
DCMRFYJHLUULFD
|
6.2 | Ki | 2 | — | |
PVLAODDTBSTRJQ
|
6.1 | Ki | 2 | — | |
BECPDRSBQZULOY
|
6.1 | Ki | 2 | — | |
KFIPPTVKFZQMJH
|
6.1 | Ki | 2 | — | |
ZVGFUPSZBYCCIH
|
6.1 | IC50 | 2 | — | |
NYUCDBAHTJBQSP
|
6.1 | Ki | 2 | — | |
LDHKTVULLKPADL
|
6.0 | IC50 | 3 | — | |
RFTSSZJZXOSICM
|
6.0 | Ki | 5 | — |