Target Details
| UniProt AC | Q92918 |
|---|---|
| Gene Symbol | MAP4K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00780 (CNH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 225
- Clinical molecules 20
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (225)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVAFKWRLBOEKGD
|
6.3 | IC50 | 2 | — | |
UDXKFAUNOZOTGY
|
6.3 | IC50 | 2 | — | |
URHHGZRDZIHONJ
|
6.3 | IC50 | 2 | — | |
VDXDEJQPELHSLU
|
6.3 | IC50 | 2 | — | |
VKZVWMJENMIADE
|
6.3 | IC50 | 2 | — | |
WGAUJZUEMJFDBD
|
6.3 | IC50 | 2 | — | |
WNDNOSDBRCNUAW
|
6.3 | IC50 | 2 | — | |
WYQOOVPHNNJHMZ
|
6.3 | IC50 | 2 | — | |
YJWAUBCYDYZIIG
|
6.3 | IC50 | 2 | — | |
ZFEUOGPGKMODOZ
|
6.3 | IC50 | 2 | — | |
ZFIOIMARIIJADT
|
6.3 | IC50 | 2 | — | |
ZUMUKHVVDXACCJ
|
6.3 | IC50 | 2 | — | |
ZYSYOACDZZDUSZ
|
6.3 | IC50 | 2 | — | |
ZZGXBFJZLKCYOO
|
6.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
6.2 | Kd | 92 | — | |
CUIHSIWYWATEQL
|
6.1 | Kd | 61 | Yes | |
PHXJVRSECIGDHY
|
6.1 | Kd | 59 | — | |
MPVGZUGXCQEXTM
|
6.1 | Kd | 61 | Yes | |
FLBNLJLONKAPLR
|
6.1 | Kd | 31 | — | |
HHZIURLSWUIHRB
|
6.0 | Kd | 57 | Yes | |
XXJWYDDUDKYVKI
|
6.0 | Kd | 52 | — | |
ZBNZXTGUTAYRHI
|
6.0 | Kd | 102 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |